January 2021
- Rietmeyer, N. Fix-boulier, C. Le Fournis, L. Iannazzo, C. Kitoun, D. Patin, D. Mengin-lecreulx, M. Etheve-Quelquejeu, M. Arthur, M. Fonvielle “Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus”, Nucleic Acid Res. 2021, Accepted. DOI: http://doi.org/10.1093/nar/gkaa1242
- S. Saidjalolov, Z. Edoo, M. Fonvielle, L. Mayer, L. Iannazzo, M. Arthur, M. Etheve-Quelquejeu, E. Braud “Synthesis of carbapenems containing peptidoglycan-mimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity” Chem. Eur. J., 2021, Accepted. DOI: http://doi.org/10.1002/chem.202004831
November 2020
- B. Li, Y. Li, C. Tomkiewicz-Raulet, P. Dao, D. Lietha, E. Yen-Pon, Z. Du, X. Coumoul, C. Garbay, M. Etheve-Quelquejeu, H. Chen “Design, Synthesis, and Biological Evaluation of Covalent Inhibitors of Focal Adhesion Kinase (FAK) against Human Malignant Glioblastoma” J. Med. Chem. 2020, 63, 12707-12724. DOI: 10.1021/acs.jmedchem.0c01059
- M. Bosco, S.-J. Paik, P. Busca, S. E. H. Moore, C. Gravier-Pelletier “Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation” Molecules 2020, 25, 4969. DOI: 10.3390/molecules25214969
- C. Fleurisson, E. Benedetti, L. Micouin Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications Synlett published online. DOI: 10.1055/s-0040-1707324
- X. Chen, P. Coric, V. Larue, S. Turcaud, X. Wang, S. Nonin-Lecomte, S. Bouaziz “The HIV-1 maturation inhibitor, EP39, interferes with the dynamic helix-coil equilibrium of the CA-SP1 junction of Gag” Eur. J. Med. Chem., 2020, 204, 112634 DOI: https://doi.org/10.1016/j.ejmech.2020.112634
October 2020
- C. Kitoun, M. Fonvielle, N. Sakkas, M. Lefresne, F. Djago, Q. Blancart Remaury, P. Poinot, M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo. “Phosphine-Mediated Bioconjugation of the 3′-end of RNA” Org. Lett., 2020, Just Acccepted. https://doi.org/10.1021/acs.orglett.0c02982
- C. Aubry, P. Clerici, C. Gerbaud, L. Micouin, J.-L. Pernodet, S. Lautru, Revised structure of Anthelvencine A and characterization of the Anthelvencin Biosynthetic gene cluster. ACS Chem Biol. 2020, 15, 945-951. https://doi.org/10.1021/acschembio.9b00960
- T. Zhang, L. Le Corre, O. Reinaud, B. Colasson “A Promising Approach for Controlling the 2nd Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen-Bonded Capsule” Chem. Eur. J. 2020 in press. https://doi.org/10.1002/chem.202004370.
- J. K. Aw, K. C. Boellaard, T. K. Tan, J. Yap, Y.P. Loh, B. Colasson, È. Blanc, Y. Lam, F. M. Fung “Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App” J. Chem. Ed. 2020, 97, 3877-3881. https://doi.org/10.1021/acs.jchemed.0c00387
July 2020
2) H.Liu, Ping Yi, W. Zhao, Y. Wu, F. Acher, J.-P. Pin, J. Liu and P. Rondard “Illuminating the allosteric modulation of the calcium-sensing receptor” PNAS Just Accepted article
3) C. Atdjian, D. Coelho, L. Iannazzo , M. Ethève-Quelquejeu, E. Braud “Synthesis of Triazole-Linked SAM-Adenosine Conjugates: Functionalization of Adenosine at N-1 or N-6 Position without Protecting Groups” Molecules 2020, 25, 3241; https://doi.org/10.3390/molecules25143241
Mai 2020
April 2020
March 2020
(2) Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, Giros B, Epelbaum J, Rosenmund C, Dutar P, Daumas S, El Mestikawy S, Pietrancosta N. “LSP5-2157 a new inhibitor of vesicular glutamate transporters.” Neuropharmacology. 2020 164 107902. doi: 10.1016/j.neuropharm.2019.
January 2020
October 2019
November 2019
December 2019
- H. Habrian, J. Levitz, V. Vyklicky, Z. Fu, A.Hoagland, I. McCort-Tranchepain, F. Acher, E. Y. Isacoff “Conformational pathway provides unique sensitivity to a synaptic mGluR” Nature Commun. 2019, 10, 5572 doi:10.1038/s41467-019-13407-8
- Abi Fayssal, A. Giungi, F. Berhal, G. Prestat “Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes” Org. Process Res. Dev., 10.1021/acs.oprd.9b00400