Mars 2024

 

  1. D. Coelho, Y. Colas, M. Etheve-Quelquejeu, E. Braud, L. Iannazzo “Halo-1,2,3-triazole: valuable compounds to access biologically relevant molecules” ChemBioChem 2024doi.org/10.1002/cbic.202400150
February 2024

 

  1. T. Zhao, E. Sachon, L. Micouin, R. Piccardi α-Silylated Diazoalkynes: New Tools for Bioconjugation of Proteins” 2024, just accepted.
    DOI: 10.1002/chem.202302807
November 2023

 

  1. Corbeski, P. Andrés Vargas-Rosales, R. Kumar Bedi, J. Deng, D. Coelho, E. Braud, L. Iannazzo, Y. Li, D. Huang, M. Ethève-Quelquejeu, Q. Cui, A. Caflisch “The catalytic mechanism of the RNA-methyltransferase METTL3”, eLife, 2023, 12:RP92537 DOI:10.7554/eLife.92537.1
  2. Brom, J.; Maruani, A.; Turcaud, S.; Lajnef, S.; Peyrot, F.; Micouin, L.; Benedetti, E. “[2.2]Paracyclophane-based coumarins: effective organo-photocatalysts for light-induced desulfonylation processes” Org. Biomol. Chem. 2023, just accepted. DOI: 10.1039/D3OB01711G (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2023-n4ds3).
September 2023

 

  1. Polikanov, Y.S, Etheve-Quelquejeu, Micura R. M. “Synthesis of Peptidyl-tRNA Mimics for Structural Biology Applications” Accounts of Chemical Research, 2023, doi-org.ezproxy.u-paris.fr/10.1021.
Mai 2023

 

  1. Le Corre L., Padovani D. “Mechanism-based and computational modeling of hydrogen sulfide biogenesis inhibition: interfacial inhibition” Scientific reports, 2023, 13, 7287. Doi: https://www.nature.com/articles/s41598-023-34405-3
  2. Coelho, D.; Le Corre, L.; Bartosik, K.; Iannazzo, L.; Braud, E.; Etheve-Quelquejeu, M. “Synthesis of Bisubstrate Analogues for RNA Methylation Studies using two Transition Metal-Catalyzed Reactions” Chem. Eur. J. 2023, e202301134.
April 2023
  1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
  2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
February 2023
  1. Flavie Bouchet, Jean-Philippe Barnier, Ines Sayah, Youcef Bagdad, Maria A. Miteva, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Ruthenium-Catalyzed Cycloaddition for Introducing Chemical Di-versity in Second generation b-Lactamase inhibitors”. ChemMedChem 2023, e202300077.
  2. Rančić A., Babić N., Orio M., Peyrot F. “Structural Features Governing the Metabolic Stability of Tetraethyl-Substituted Nitroxides in Rat Liver Microsomes”  Antioxidants, 2023, 12(2), 402. DOI:  https://doi.org/10.3390/antiox12020402
January 2023
  1. Felder, S.; Delcourt, M.-L.; Rodríguez, R.; Favereau, L.; Jeanne Crassous, J.; Micouin, L.; Benedetti, E. “Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives”, J. Mater. Chem. C 202311, 2053 DOI: https://doi.org/10.1039/D2TC04885J
  2. Galardon, E.; Mathas, N.; Padovani, D.; Le Corre, L.; Poncet, G.; Dairou, J. Persulfidation of DJ-1: Mechanism and Consequences.” Biomolecules 2023, 13, 27. DOI: https://doi.org/10.3390/biom13010027
December 2022
  1. Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein “Enzymatic synthesis of vancomycin-modified DNA”, Molecule, 2022, doi.org/10.3390/molecules27248927
October 2022
  1. C. Kitoun, S. Saidjalolov, D. Bouquet, F. Djago, Q. Blancart Remaury, B. Sargueil, P. Poinot, Pauline; M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger Ligation to Access to Stable Aminoacyl- or Peptidyl-dinucleotides” ACS Omega., 2022, just accepted.
  2. Rietmeyer, L.; Li de la Sierra-Gallay, I.; Schepers, G.; Dorchêne, D.; Iannazzo, L.; Patin, D.; Touzé, T.; van Tilbeurgh, H.; Herdewijn, P.; Etheve-Quelquejeu, M.; Fonvielle, M. “Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis” Nucleic Acids Research, 2022, just accepted
  3. S. Felder, C. Sagné, E. Benedetti, L. Micouin “Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity
    through Scaffold Hopping” ACS Chemical Biology, 2022, 17, 3069. DOI: https://doi.org/10.1021/acschembio.2c00171
August 2022

1) J.-P. Barnier, S. Saidjalolov, F. Bouchet, L. Mayer, Z. Edoo, I. Sayah, L. Iannazzo, M.e Ethève-Quelquejeu, J.-L. Mainardi, E. Braud “Modulation of the Specificity of Carbapenems and Diazabicyclooctanes for Selective Activity against Mycobacterium tuberculosis” Antimicrob. Agents Chemother. 2022, Ahead of Print

DOI: https://doi.org/10.1128/aac.02357-21

June 2022

1) F. Peyrot, S. Lajnef, D.-L. Versace. “Electron Paramagnetic Resonance Spin Trapping (EPR–ST) Technique in Photopolymerization Processes” Catalysts, 2022, 12, (7), 772; DOI: https://doi.org/10.3390/catal12070772

Mai 2022

1) V. Meynier, L. Iannazzo, M. Catala, S. Oerum, E. Braud, C.Atdjian, P. Barraud, M. Fonvielle, C. Tisné, M.Ethève-Quelquejeu “Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase” Nucleic Acids Research, 2022, 50, (10), 5793–5806. DOI: https://doi.org/10.1093/nar/gkac354

April 2022
  1. M. F. Cunha,   I.Pranke, A. Sassi, C. Schreiweis, S.  Moriceau, D. Vidovic, A. Hatton, M. S. Carlon, G. Creste, F. Berhal, G. Prestat, R. Freund, N. Odolczyk, J. P. Jais, C. Gravier-Pelletier, P.  Zielenkiewicz, V. Jullien, A. Hinzpeter, F. Oury, A. Edelman, I. Sermet-Gaudelus “Systemic Bis-Phosphinic Acid Derivative Restores Chloride Transport in Cystic Fibrosis Mice” Sci Rep 2022, 12 (1), 6132. DOI: https://doi.org/10.1038/s41598-022-09678-9.
  2. Li, K. Aubertin, D. Onidas, P. Nizard, N. Felidj, F. Gazeau, C. Mangeney, Y. Luo “Recent advances in non-plasmonic SERS nanostructures for biomedical applications” WIREs Nanomedicine & Nanobiotechnology 2022. DOI: https://doi.org/10.1002/wnan.1795
Mars 2022

1) M. Oliver, L, Le Corre, M. Poinsot, M, Bosco, H. Wan, A. Amoroso, B. Joris, A. Bouhss, S. Calvet-Vitale, C. Gravier-Pelletier “A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling” Molecules 2022, 27(6), 1769. DOI:  https://doi.org/10.3390/molecules27061769

February 2022
  1. D. Padovani, E. Galardon, “Molecular Basis for the Interaction of Catalase with d-Penicillamine: Rationalization of Some of Its Deleterious Effects” Chem. Res. Toxicol. 2022, 35, 3, 412–421 DOI: https://doi.org/10.1021/acs.chemrestox.1c00313
Janaury 2022
  1. D. R. Boyd, N. D. Sharma, P. J. Stevenson, P. Hoering, C. C. R. Allen, P. M. Dansette “Monooxygenase- and Dioxygenase-Catalyzed Oxidative Dearomatization of Thiophenes by Sulfoxidation, cis-Dihydroxylation and Epoxidation”. Int J Mol Sci. 2022, 23(2) 909. DOI:https://doi.org/10.3390/ijms23020909 
  2. Li, P. Nizard, D. Onidas, A. Lamouri, J. Pinson, S. Mahouche-Chergui, K. Aubertin, F. Gazeau, Y. Luo, C. Mangeney “SERS Tags Derived from Silver Nanoparticles and Aryl Diazonium Salts for Cell Raman Imaging” Nanoscale 2022, 14, 1452. DOI: https://doi.org/10.1039/D1NR03148A
  3. Bicyclic 5-5 systems with one ring junction nitrogen atom: Two extra heteroatoms 2:0 Benedetti, E.; Micouin, L. Reference Collection in Chemistry, Molecular Science and Chemical Engineering Wiley, 2022. Volume 11, pp 145-173. DOI:10.1016/B978-0-12-409547-2.14935-2 
December 2021
  1. S. Felder, M.-L. Delcourt, M.H.E. Bousquet, D.  Jacquemin, R. Rodríguez, L. Favereau, J. Crassous, L. Micouin, E. Benedetti “Planar chiral analogues of PRODAN based on a [2.2]paracyclophane scaffold: Synthesis and photophysical studies”. J. Org. Chem. 2021, just accepted
  2. G. Kirby, L. Grimaud, M. R. Vitale,  G. Prestat, F. Berhal “Iron(ii)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources” Green Chem., 2021,23, 9428-9432. https://doi.org/10.1039/D1GC03495B
  3. G. De Leener, D. Over, O. Reinaud, I. Jabin Turning on anion and betaine hosting by a small structural change of a biomimetic cavity: a case study” Supramol. Chem. 2021, DOI: 10.1080/10610278.2021.2011890
  4. Bitam, S.; Elbahnsi, A.; Creste, G.; Pranke, I.; Chevalier, B.; Berhal, F.; Hoffmann, B.; Servel, N.; Tondelier, D.; Hatton, A.; Moquereau, C.; Faria Da Cunha, M.; Pastor, A.; Lepissier, A.; Hinzpeter, A.; Mornon, J.-P.; Prestat, G.; Edelman, A.; Callebaut, I.; Gravier-Pelletier, C.; Sermet-Gaudelus, I. “New Insights into Structure and Function of Bis-Phosphinic Acid Derivatives and Implications for CFTR Modulation.” Sci Rep 2021, 11, 6842.
    DOI: https://doi.org/10.1038/s41598-021-83240-x
  5. Bardin, E.; Pastor, A.; Semeraro, M.; Golec, A.; Hayes, K.; Chevalier, B.; Berhal, F.; Prestat, G.; Hinzpeter, A.; Gravier-Pelletier, C.; Pranke, I.; Sermet-Gaudelus, I. “Modulators of CFTR. Updates on Clinical Development and Future Directions.” Eur. J. Med. Chem. 2021, 113195  DOI: doi.org/10.1016/j.ejmech.2021.113195
  6. Oliver, M.; Le Corre, L.; Poinsot, M.; Corio, A.; Madegard, L.; Bosco, M.; Amoroso, A.; Joris, B.; Auger, R.; Touzé, T.; Bouhss, A.; Calvet-Vitale, S.; Gravier-Pelletier, C.“Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors.”  Org. Biomol. Chem. 2021, 19(26), 5844-5866, DOI: 10.1039/D1OB00710F.
  7. Pujol C, Legrand A, Parodi L, Boucher, J.-L.; Le Corre, L. et al. “Implication of folate deficiency in CYP2U1 loss of function.” J Exp Med. 2021; 218(11):e20210846. doi: 10.1084/jem.20210846.
October 2021
  1. S. Wu, L.A. Galan, M. Roux, F. Riobe, B. Le Guennic, Y. Guyot, T. Le Bahers, L. Micouin, O. Maury, E. Benedetti “Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation” Inorg. Chem. 2021, 60, 16194−16203. DOI: https://doi.org/10.1021/acs.inorgchem.1c01986.
  2. F. Bouchet, H. Atze,  M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger ligation to introduce chemical diversity on β-lactamase inhibitors of second generation” Org. Lett.2021, just accepted
  3. Médard, X. Sun, J. Pinson, D. Li, C. Mangeney, J.-P. Michel “Electrografting and Langmuir-Blodgett: Covalently Bound Nanometer Thick Ordered Films on Graphite” Langmuir 2021, 37, 12539. DOI: https://doi.org/10.1021/acs.langmuir.1c01723
September 2021
​A. Corio, C. Gravier-Pelletier, P. Busca “Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review.” Molecules 2021, 26(18), 5467. DOI: https://doi.org/10.3390/molecules26185467
August 2021
  1. ​J. Haubrich, J. Font, R. B. Quast, A. Goupil-Lamy, P. Scholler, D. Nevoltris, F.Acher, P. Chames, P. Rondard, L. Prezeau, J.-P. Pin “A nanobody activating metabotropic glutamate receptor 4 discriminates between homo and heterodimers.” Proc. Natl. Acad. Sci. U S A 2021,
  2. Li, Y. Luo, D. Onidas, L. He, M. Jin, F. Gazeau, J. Pinson, C. Mangeney “Surface functionalization of nanomaterials by aryl diazonium salts for biomedical sciences” Adv. Colloid & Interface Science 2021, 294, 102479. DOI: https://doi.org/10.1016/j.cis.2021.102479
July 2021
  1. Xiao, J. Gateau, A. Brun, X. Shi, F. Gazeau, C. Mangeney, Y. Luo “Hybrid nano- and microgels doped with photoacoustic contrast agents for cancer theranostics” View 2021, 2:20200176. DOI: https://doi.org/10.1002/VIW.20200176
June 2021
  1. S. Felder, S. Wu, J. Brom, L. Micouin, E. Benedetti Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis”  Chirality, 2021, 33, 506-527 DOI: https://doi.org/10.1002/chir.23335
Mai 2021
  1. Kherbouche, D. McRae, T. Geronimi, F. Lagugné-Labarthet, A. Lamouri, A. Chevillot-Biraud, C. Mangeney, N. Felidj “Extending nanoscale patterning with multipolar surface plasmon resonances” Nanoscale 2021, 13, 11051. DOI: https://doi.org/10.1039/D1NR02181H
Mars 2021
  1. S. Felder, L. Micouin, E. Benedetti “Para‐functionalization of N‐substituted 4‐amino[2.2]paracyclophanes by regioselective formylation” Eur. J. Org. Chem., 2021, 4015-4018. DOI: https://doi.org/10.1002/ejoc.202100288
  2. Barosi, A. Berisha, C. Mangeney, J. Pinson, H. Dhimane, P. I. Dalko “Efficient construction of redox responsive thin polymer layer on carbon and gold for voltage-gated delivery applications” Materials Adv. 2021, 2, 2358. DOI: https://doi.org/10.1039/D1MA00022E
February 2021
  1. D.A.B. Therien, D. M. McRae, C. Mangeney, N. Félidj, F. Lagugné-Labarthet “Three-Color Plasmon-Mediated Reduction of Diazonium Salts over Metasurfaces” Nanoscale Adv. 2021, 3, 2501. DOI: https://doi.org/10.1039/D0NA00862A

January 2021
  1. Rietmeyer, N. Fix-boulier, C. Le Fournis, L. Iannazzo, C. Kitoun, D. Patin, D. Mengin-lecreulx, M. Etheve-Quelquejeu, M. Arthur, M. Fonvielle “Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus”, Nucleic Acid Res. 2021, Accepted. DOI: http://doi.org/10.1093/nar/gkaa1242
  2. S. Saidjalolov, Z. Edoo, M. Fonvielle, L. Mayer, L. Iannazzo, M. Arthur, M. Etheve-Quelquejeu, E. Braud “Synthesis of carbapenems containing peptidoglycan-mimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity” Chem. Eur. J., 2021, Accepted. DOI: http://doi.org/10.1002/chem.202004831
  3. de Sa Nogueira D, Bourdy R, Filliol D, Quessada C, McCort-Tranchepain I, Acher F, Zwiller J, Romieu P, Befort K. “LSP2-9166, an orthosteric mGlu4 and mGlu7 receptor agonist, reduces cocaine self-administration under a progressive ratio schedule in rats” Neurosci Lett. 2020, 135603 https://doi.org/10.1016/j.neulet.2020.135603
  4. K. Abbas, N. Babić, F. Peyrot. “Detection of superoxide radical in adherent living cells by electron paramagnetic resonance (EPR) spectroscopy using cyclic nitrones”. Methods Mol. Biol. 2021, 2202, 149-163. DOI: https://doi.org/10.1007/978-1-0716-0896-8_13
November 2020
  1. B. Li, Y. Li, C. Tomkiewicz-Raulet, P. Dao, D. Lietha, E. Yen-Pon, Z. Du, X. Coumoul, C. Garbay, M. Etheve-Quelquejeu, H. Chen “Design, Synthesis, and Biological Evaluation of Covalent Inhibitors of Focal Adhesion Kinase (FAK) against Human Malignant Glioblastoma” J. Med. Chem. 202063, 12707-12724. DOI: 10.1021/acs.jmedchem.0c01059
  2. M. Bosco, S.-J. Paik, P. Busca, S. E. H. Moore, C. Gravier-Pelletier “Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation” Molecules 2020, 25, 4969. DOI: 10.3390/molecules25214969
  3. C. Fleurisson, E. Benedetti, L. Micouin Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications Synlett 2021, 31, 858-874. DOI: 10.1055/s-0040-1707324
  4. X. Chen, P. Coric, V. Larue, S. Turcaud, X. Wang, S. Nonin-Lecomte, S. Bouaziz “The HIV-1 maturation inhibitor, EP39, interferes with the dynamic helix-coil equilibrium of the CA-SP1 junction of Gag” Eur. J. Med. Chem.2020204, 112634 DOI: https://doi.org/10.1016/j.ejmech.2020.112634
October 2020
  1. C. Kitoun, M. Fonvielle, N. Sakkas, M. Lefresne, F. Djago, Q. Blancart Remaury, P. Poinot, M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo. “Phosphine-Mediated Bioconjugation of the 3′-end of RNA” Org. Lett., 2020, Just Acccepted.   https://doi.org/10.1021/acs.orglett.0c02982
  2. C. Aubry, P. Clerici, C. Gerbaud, L. Micouin, J.-L. Pernodet, S. Lautru, Revised structure of Anthelvencine A and characterization of the Anthelvencin Biosynthetic gene cluster.  ACS Chem Biol. 2020, 15, 945-951. https://doi.org/10.1021/acschembio.9b00960
  3. T. Zhang, L. Le Corre, O. Reinaud, B. Colasson “A Promising Approach for Controlling the 2nd Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen-Bonded Capsule” Chem. Eur. J. 2020 in press. https://doi.org/10.1002/chem.202004370.
  4. J. K. Aw, K. C. Boellaard, T. K. Tan, J. Yap, Y.P. Loh, B. Colasson, È. Blanc, Y. Lam, F. M. Fung “Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App” J. Chem. Ed. 2020, 97, 3877-3881. https://doi.org/10.1021/acs.jchemed.0c00387
July 2020
1) Dubois L, Pietrancosta N, Cabaye A, Fanget I, Debacker C, Gilormini PA, Dansette PM, Dairou J, Biot C, Froissart R, Goupil-Lamy A, Bertrand HO, Acher FC, McCort-Tranchepain I, Gasnier B, Anne C. “Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin.” J. Med. Chem. 2020  Online ahead of print.  https://doi.org/10.1021/acs.jmedchem.9b02119.  PMID: 32608236

2) H.Liu, Ping Yi, W. Zhao, Y. Wu, F. Acher, J.-P. Pin, J. Liu and P. Rondard “Illuminating the allosteric modulation of the calcium-sensing receptor” Proc Natl Acad Sci U S A 2020, 117, 21711-21722. https://doi.org/10.1073/pnas.1922231117

3) C. Atdjian, D. Coelho, L. Iannazzo , M. Ethève-Quelquejeu, E. Braud “Synthesis of Triazole-Linked SAM-Adenosine Conjugates: Functionalization of Adenosine at N-1 or N-6 Position without Protecting Groups” Molecules 2020, 25, 3241; https://doi.org/10.3390/molecules25143241

June 2020
  1. N. Babić, M. Orio, F. Peyrot. “Unexpected rapid aerobic transformation of 2,2,6,6-tetraethyl-4-oxo(piperidin-1-yloxyl) radical by cytochrome P450 in the presence of NADPH: Evidence against a simple reduction of the nitroxide moiety to the hydroxylamine”. Free Radic. Biol. Med. 2020, 156, 144-156. DOI: https://doi.org/10.1016/j.freeradbiomed.2020.05.021
  2. Kherbouche, Y. Luo, N. Félidj, C. Mangeney “Plasmon-Mediated Surface Functionalization: New Horizons for the Control of Surface Chemistry on the Nanoscale” Chem. Mater. 2020, 32, 5442. DOI: https://doi.org/10.1021/acs.chemmater.0c00921

 

Mai 2020
  1. Y. LuoY. XiaoD. OnidasL. IannazzoM. Ethève-QuelquejeuA. LamouriN. FélidjS. Mahouche-CherguiT. BruléN. Gagey-EilsteinF. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles”.  Chem. Commun., 2020, Advance Article https://doi.org/10.1039/D0CC02842H
  2. Decorbie, I. Tijunelyte, S. Gam-Derouich, J. Solard, A. Lamouri, P. Decorse, N. Felidj, C. Gauchotte-Lindsay, E. Rinnert, C. Mangeney, N. Lidgi-Guigui “Sensing Polymer/Paracetamol Interaction with an Independent Component Analysis-Based SERS-MIP Nanosensor” Plasmonics 2020, 15, 1533. DOI: https://doi.org/10.1007/s11468-020-01177-9
  3. Luo, Y. Xiao, D. Onidas, L. Iannazzo, M. Ethève-Quelquejeu, A. Lamouri, N. Félidj, S. Mahouche-Chergui, T. Brulé, N. Gagey-Eilstein, F. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles” Chem. Commun. 2020, 56, 6822. DOI: https://doi.org/10.1039/D0CC02842H
April 2020
(1) Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Diazabicyclooctane functionalization for inhibition of β-lactamases from enterobacteria”. Journal of Medicinal Chemistry, Just Accepted, https://doi.org/10.1021/acs.jmedchem.9b02125
March 2020
(1) A. Mikou, A. Cabayé, A. Goupil, H.-O. Bertrand, J.-P. Mothet, F. Acher “Asc-1 Transporter (SLC7A10): Homology models and molecular dynamics insights into the first steps of the transport mechanism.” Sci.Rep. DOI: doi.org/10.1038/s41598-020-60617-y

(2) Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, Giros B, Epelbaum J, Rosenmund C, Dutar P, Daumas S, El Mestikawy S, Pietrancosta N. “LSP5-2157 a new inhibitor of vesicular glutamate transporters.” Neuropharmacology. 2020 164 107902. doi: 10.1016/j.neuropharm.2019.107902.

January 2020
  1. Médard, P. Decorse, C. Mangeney, J. Pinson, M. Fagnoni, S. Protti “Simultaneous Photografting of Two Organic Groups on a Gold Surface by using Arylazo Sulfones as Single Precursors” Langmuir 2020, 36, 11, 2786. DOI: https://doi.org/10.1021/acs.langmuir.9b03878

 

January 2020
B. Colasson, A. Credi, B. Ventura “Photoinduced electron transfer involving a naphthalimide chromophore in switchable and flexible [2]rotaxanes“ Chem. Eur. J.202026, 534-542. doi: 10.1002/chem.201904155.
December 2019
  1. H. Habrian, J. Levitz, V. Vyklicky, Z. Fu, A.Hoagland, I. McCort-Tranchepain, F. Acher, E. Y. Isacoff “Conformational pathway provides unique sensitivity to a synaptic mGluR” Nature Commun. 2019, 10, 5572 doi:10.1038/s41467-019-13407-8
  2. Abi Fayssal, A. Giungi, F. Berhal, G. Prestat “Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes” Org. Process Res. Dev., 10.1021/acs.oprd.9b00400
November 2019
Hayek, N. Pietrancosta, A. A. Hovhannisyan, R. Alves de Sousa N. Bekaddour, L. Ermellino, E. Tramontano, S. Arnould, C. Sardet, J. Dairou, O. Diaz, V. Lotteau, S. Nisole, G. Melikyan, J.-H. Herbeuval, P.- O. Vidalain. “Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition” Eur. J. Med. Chem. DOI: 10.1016/j.ejmech.2019.111855
October 2019
Zahim, D. Ajami, P. Laurent, H. Valkenier, O. Reinaud, M. Luhmer, I. Jabin ” Synthesis and Binding Properties of a Tren-Capped Hexahomotrioxacalix[3]arene” ChemPhysChem 10.1002/cphc.201900951
September 2019

N. Babić, F. Peyrot. “New synthetic route to 2,2,6,6-tetraethylpiperidin-4-one: A key-intermediate towards tetraethyl nitroxides”. Tet. Lett. 2019, 60(44), 151207. DOI: https://doi.org/10.1016/j.tetlet.2019.151207

February 2019

N. Babić, F. Peyrot. “Molecular Probes for Evaluation of Oxidative Stress by In Vivo EPR Spectroscopy and Imaging: State-of-the-Art and Limitations”. Magnetochemistry 2019, I(1), 13. DOI: https://doi.org/10.3390/magnetochemistry5010013

june 2023

 

  1. Moreau TRJ., Bondet V., Rodero MP., Duffy D. “Heterogeneity and functions of the 13 IFN-α subtypes – lucky for some?” Eur J Immunol. 2023 Jun 27:e2250307. doi: 10.1002/eji.202250307.
  2. Fayand A., Hentgen V., Posseme C., Lacout C., Picard C., Moguelet P., Cescato M., Sbeih N., Moreau TRJ., Zhu YY., Charuel JL., Corneau A., Deibener-Kaminsky J., Dupuy S., Fusaro M., Hoareau B., Hovnanian A., Langlois V., Le Corre L., Maciel TT., Miskinyte S., Miyara M., Moulinet T., Perret M., Schuhmacher MH., Rignault-Bricard R., Viel S., Vinit A., Soria A., Duffy D., Launay JM., Callebert J., Herbeuval JP., Rodero MP., Georgin-Lavialle S. “Successful treatment of JAK1 associated inflammatory disease.” J Allergy Clin Immunol. 2023 Jun 19:S0091-6749(23)00799-6. doi: 10.1016/j.jaci.2023.06.004
  3. Bader-Meunier B., Breton S., Duffy D., Gitiaux C., Quartier P., Lemelle I., Meyer A., Welfringer-Morin A., Frémond ML., Charuel JL., Rodero MP., Melki I. “Osteonecrosis in patients with juvenile dermatomyositis: is it associated with anti-MDA5 autoantibody?” Rheumatology (Oxford). 2023 Jan 2:keac696. doi: 10.1093/rheumatology/keac696.
Mai 2023

 

  1. Le Corre L., Padovani D. “Mechanism-based and computational modeling of hydrogen sulfide biogenesis inhibition: interfacial inhibition” Scientific reports, 2023, 13, 7287. Doi: https://www.nature.com/articles/s41598-023-34405-3
  2. Coelho, D.; Le Corre, L.; Bartosik, K.; Iannazzo, L.; Braud, E.; Etheve-Quelquejeu, M. “Synthesis of Bisubstrate Analogues for RNA Methylation Studies using two Transition Metal-Catalyzed Reactions” Chem. Eur. J. 2023, e202301134.
April 2023
  1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
  2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
February 2023
  1. Flavie Bouchet, Jean-Philippe Barnier, Ines Sayah, Youcef Bagdad, Maria A. Miteva, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Ruthenium-Catalyzed Cycloaddition for Introducing Chemical Di-versity in Second generation b-Lactamase inhibitors”. ChemMedChem 2023, e202300077.
  2. Rančić A., Babić N., Orio M., Peyrot F. “Structural Features Governing the Metabolic Stability of Tetraethyl-Substituted Nitroxides in Rat Liver Microsomes”  Antioxidants, 2023, 12(2), 402. DOI:  https://doi.org/10.3390/antiox12020402
January 2023
  1. Felder, S.; Delcourt, M.-L.; Rodríguez, R.; Favereau, L.; Jeanne Crassous, J.; Micouin, L.; Benedetti, E. “Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives”, J. Mater. Chem. C 202311, 2053 DOI: https://doi.org/10.1039/D2TC04885J
  2. Galardon, E.; Mathas, N.; Padovani, D.; Le Corre, L.; Poncet, G.; Dairou, J. Persulfidation of DJ-1: Mechanism and Consequences.” Biomolecules 2023, 13, 27. DOI: https://doi.org/10.3390/biom13010027
December 2022
  1. Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein “Enzymatic synthesis of vancomycin-modified DNA”, Molecule, 2022, doi.org/10.3390/molecules27248927
October 2022
  1. C. Kitoun, S. Saidjalolov, D. Bouquet, F. Djago, Q. Blancart Remaury, B. Sargueil, P. Poinot, Pauline; M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger Ligation to Access to Stable Aminoacyl- or Peptidyl-dinucleotides” ACS Omega., 2022, just accepted.
  2. Rietmeyer, L.; Li de la Sierra-Gallay, I.; Schepers, G.; Dorchêne, D.; Iannazzo, L.; Patin, D.; Touzé, T.; van Tilbeurgh, H.; Herdewijn, P.; Etheve-Quelquejeu, M.; Fonvielle, M. “Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis” Nucleic Acids Research, 2022, just accepted
  3. S. Felder, C. Sagné, E. Benedetti, L. Micouin “Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity
    through Scaffold Hopping” ACS Chemical Biology, 2022, 17, 3069. DOI: https://doi.org/10.1021/acschembio.2c00171
August 2022

1) J.-P. Barnier, S. Saidjalolov, F. Bouchet, L. Mayer, Z. Edoo, I. Sayah, L. Iannazzo, M.e Ethève-Quelquejeu, J.-L. Mainardi, E. Braud “Modulation of the Specificity of Carbapenems and Diazabicyclooctanes for Selective Activity against Mycobacterium tuberculosis” Antimicrob. Agents Chemother. 2022, Ahead of Print

DOI: https://doi.org/10.1128/aac.02357-21

June 2022

1) F. Peyrot, S. Lajnef, D.-L. Versace. “Electron Paramagnetic Resonance Spin Trapping (EPR–ST) Technique in Photopolymerization Processes” Catalysts, 2022, 12, (7), 772; DOI: https://doi.org/10.3390/catal12070772

Mai 2022

1) V. Meynier, L. Iannazzo, M. Catala, S. Oerum, E. Braud, C.Atdjian, P. Barraud, M. Fonvielle, C. Tisné, M.Ethève-Quelquejeu “Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase” Nucleic Acids Research, 2022, 50, (10), 5793–5806. DOI: https://doi.org/10.1093/nar/gkac354

April 2022
  1. M. F. Cunha,   I.Pranke, A. Sassi, C. Schreiweis, S.  Moriceau, D. Vidovic, A. Hatton, M. S. Carlon, G. Creste, F. Berhal, G. Prestat, R. Freund, N. Odolczyk, J. P. Jais, C. Gravier-Pelletier, P.  Zielenkiewicz, V. Jullien, A. Hinzpeter, F. Oury, A. Edelman, I. Sermet-Gaudelus “Systemic Bis-Phosphinic Acid Derivative Restores Chloride Transport in Cystic Fibrosis Mice” Sci Rep 2022, 12 (1), 6132. DOI: https://doi.org/10.1038/s41598-022-09678-9.
  2. Li, K. Aubertin, D. Onidas, P. Nizard, N. Felidj, F. Gazeau, C. Mangeney, Y. Luo “Recent advances in non-plasmonic SERS nanostructures for biomedical applications” WIREs Nanomedicine & Nanobiotechnology 2022. DOI: https://doi.org/10.1002/wnan.1795
Mars 2022

1) M. Oliver, L, Le Corre, M. Poinsot, M, Bosco, H. Wan, A. Amoroso, B. Joris, A. Bouhss, S. Calvet-Vitale, C. Gravier-Pelletier “A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling” Molecules 2022, 27(6), 1769. DOI:  https://doi.org/10.3390/molecules27061769

February 2022
  1. D. Padovani, E. Galardon, “Molecular Basis for the Interaction of Catalase with d-Penicillamine: Rationalization of Some of Its Deleterious Effects” Chem. Res. Toxicol. 2022, 35, 3, 412–421 DOI: https://doi.org/10.1021/acs.chemrestox.1c00313
Janaury 2022
  1. D. R. Boyd, N. D. Sharma, P. J. Stevenson, P. Hoering, C. C. R. Allen, P. M. Dansette “Monooxygenase- and Dioxygenase-Catalyzed Oxidative Dearomatization of Thiophenes by Sulfoxidation, cis-Dihydroxylation and Epoxidation”. Int J Mol Sci. 2022, 23(2) 909. DOI:https://doi.org/10.3390/ijms23020909 
  2. Li, P. Nizard, D. Onidas, A. Lamouri, J. Pinson, S. Mahouche-Chergui, K. Aubertin, F. Gazeau, Y. Luo, C. Mangeney “SERS Tags Derived from Silver Nanoparticles and Aryl Diazonium Salts for Cell Raman Imaging” Nanoscale 2022, 14, 1452. DOI: https://doi.org/10.1039/D1NR03148A
  3. Bicyclic 5-5 systems with one ring junction nitrogen atom: Two extra heteroatoms 2:0 Benedetti, E.; Micouin, L. Reference Collection in Chemistry, Molecular Science and Chemical Engineering Wiley, 2022. Volume 11, pp 145-173. DOI:10.1016/B978-0-12-409547-2.14935-2 
December 2021
  1. S. Felder, M.-L. Delcourt, M.H.E. Bousquet, D.  Jacquemin, R. Rodríguez, L. Favereau, J. Crassous, L. Micouin, E. Benedetti “Planar chiral analogues of PRODAN based on a [2.2]paracyclophane scaffold: Synthesis and photophysical studies”. J. Org. Chem. 2021, just accepted
  2. G. Kirby, L. Grimaud, M. R. Vitale,  G. Prestat, F. Berhal “Iron(ii)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources” Green Chem., 2021,23, 9428-9432. https://doi.org/10.1039/D1GC03495B
  3. G. De Leener, D. Over, O. Reinaud, I. Jabin Turning on anion and betaine hosting by a small structural change of a biomimetic cavity: a case study” Supramol. Chem. 2021, DOI: 10.1080/10610278.2021.2011890
  4. Bitam, S.; Elbahnsi, A.; Creste, G.; Pranke, I.; Chevalier, B.; Berhal, F.; Hoffmann, B.; Servel, N.; Tondelier, D.; Hatton, A.; Moquereau, C.; Faria Da Cunha, M.; Pastor, A.; Lepissier, A.; Hinzpeter, A.; Mornon, J.-P.; Prestat, G.; Edelman, A.; Callebaut, I.; Gravier-Pelletier, C.; Sermet-Gaudelus, I. “New Insights into Structure and Function of Bis-Phosphinic Acid Derivatives and Implications for CFTR Modulation.” Sci Rep 2021, 11, 6842.
    DOI: https://doi.org/10.1038/s41598-021-83240-x
  5. Bardin, E.; Pastor, A.; Semeraro, M.; Golec, A.; Hayes, K.; Chevalier, B.; Berhal, F.; Prestat, G.; Hinzpeter, A.; Gravier-Pelletier, C.; Pranke, I.; Sermet-Gaudelus, I. “Modulators of CFTR. Updates on Clinical Development and Future Directions.” Eur. J. Med. Chem. 2021, 113195  DOI: doi.org/10.1016/j.ejmech.2021.113195
  6. Oliver, M.; Le Corre, L.; Poinsot, M.; Corio, A.; Madegard, L.; Bosco, M.; Amoroso, A.; Joris, B.; Auger, R.; Touzé, T.; Bouhss, A.; Calvet-Vitale, S.; Gravier-Pelletier, C.“Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors.”  Org. Biomol. Chem. 2021, 19(26), 5844-5866, DOI: 10.1039/D1OB00710F.
  7. Pujol C, Legrand A, Parodi L, Boucher, J.-L.; Le Corre, L. et al. “Implication of folate deficiency in CYP2U1 loss of function.” J Exp Med. 2021; 218(11):e20210846. doi: 10.1084/jem.20210846.
October 2021
  1. S. Wu, L.A. Galan, M. Roux, F. Riobe, B. Le Guennic, Y. Guyot, T. Le Bahers, L. Micouin, O. Maury, E. Benedetti “Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation” Inorg. Chem. 2021, 60, 16194−16203. DOI: https://doi.org/10.1021/acs.inorgchem.1c01986.
  2. F. Bouchet, H. Atze,  M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger ligation to introduce chemical diversity on β-lactamase inhibitors of second generation” Org. Lett.2021, just accepted
  3. Médard, X. Sun, J. Pinson, D. Li, C. Mangeney, J.-P. Michel “Electrografting and Langmuir-Blodgett: Covalently Bound Nanometer Thick Ordered Films on Graphite” Langmuir 2021, 37, 12539. DOI: https://doi.org/10.1021/acs.langmuir.1c01723
September 2021
​A. Corio, C. Gravier-Pelletier, P. Busca “Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review.” Molecules 2021, 26(18), 5467. DOI: https://doi.org/10.3390/molecules26185467
August 2021
  1. ​J. Haubrich, J. Font, R. B. Quast, A. Goupil-Lamy, P. Scholler, D. Nevoltris, F.Acher, P. Chames, P. Rondard, L. Prezeau, J.-P. Pin “A nanobody activating metabotropic glutamate receptor 4 discriminates between homo and heterodimers.” Proc. Natl. Acad. Sci. U S A 2021,
  2. Li, Y. Luo, D. Onidas, L. He, M. Jin, F. Gazeau, J. Pinson, C. Mangeney “Surface functionalization of nanomaterials by aryl diazonium salts for biomedical sciences” Adv. Colloid & Interface Science 2021, 294, 102479. DOI: https://doi.org/10.1016/j.cis.2021.102479
July 2021
  1. Xiao, J. Gateau, A. Brun, X. Shi, F. Gazeau, C. Mangeney, Y. Luo “Hybrid nano- and microgels doped with photoacoustic contrast agents for cancer theranostics” View 2021, 2:20200176. DOI: https://doi.org/10.1002/VIW.20200176
June 2021
  1. S. Felder, S. Wu, J. Brom, L. Micouin, E. Benedetti Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis”  Chirality, 2021, 33, 506-527 DOI: https://doi.org/10.1002/chir.23335
Mai 2021
  1. Kherbouche, D. McRae, T. Geronimi, F. Lagugné-Labarthet, A. Lamouri, A. Chevillot-Biraud, C. Mangeney, N. Felidj “Extending nanoscale patterning with multipolar surface plasmon resonances” Nanoscale 2021, 13, 11051. DOI: https://doi.org/10.1039/D1NR02181H
Mars 2021
  1. S. Felder, L. Micouin, E. Benedetti “Para‐functionalization of N‐substituted 4‐amino[2.2]paracyclophanes by regioselective formylation” Eur. J. Org. Chem., 2021, 4015-4018. DOI: https://doi.org/10.1002/ejoc.202100288
  2. Barosi, A. Berisha, C. Mangeney, J. Pinson, H. Dhimane, P. I. Dalko “Efficient construction of redox responsive thin polymer layer on carbon and gold for voltage-gated delivery applications” Materials Adv. 2021, 2, 2358. DOI: https://doi.org/10.1039/D1MA00022E
February 2021
  1. D.A.B. Therien, D. M. McRae, C. Mangeney, N. Félidj, F. Lagugné-Labarthet “Three-Color Plasmon-Mediated Reduction of Diazonium Salts over Metasurfaces” Nanoscale Adv. 2021, 3, 2501. DOI: https://doi.org/10.1039/D0NA00862A

January 2021
  1. Rietmeyer, N. Fix-boulier, C. Le Fournis, L. Iannazzo, C. Kitoun, D. Patin, D. Mengin-lecreulx, M. Etheve-Quelquejeu, M. Arthur, M. Fonvielle “Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus”, Nucleic Acid Res. 2021, Accepted. DOI: http://doi.org/10.1093/nar/gkaa1242
  2. S. Saidjalolov, Z. Edoo, M. Fonvielle, L. Mayer, L. Iannazzo, M. Arthur, M. Etheve-Quelquejeu, E. Braud “Synthesis of carbapenems containing peptidoglycan-mimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity” Chem. Eur. J., 2021, Accepted. DOI: http://doi.org/10.1002/chem.202004831
  3. de Sa Nogueira D, Bourdy R, Filliol D, Quessada C, McCort-Tranchepain I, Acher F, Zwiller J, Romieu P, Befort K. “LSP2-9166, an orthosteric mGlu4 and mGlu7 receptor agonist, reduces cocaine self-administration under a progressive ratio schedule in rats” Neurosci Lett. 2020, 135603 https://doi.org/10.1016/j.neulet.2020.135603
  4. K. Abbas, N. Babić, F. Peyrot. “Detection of superoxide radical in adherent living cells by electron paramagnetic resonance (EPR) spectroscopy using cyclic nitrones”. Methods Mol. Biol. 2021, 2202, 149-163. DOI: https://doi.org/10.1007/978-1-0716-0896-8_13
November 2020
  1. B. Li, Y. Li, C. Tomkiewicz-Raulet, P. Dao, D. Lietha, E. Yen-Pon, Z. Du, X. Coumoul, C. Garbay, M. Etheve-Quelquejeu, H. Chen “Design, Synthesis, and Biological Evaluation of Covalent Inhibitors of Focal Adhesion Kinase (FAK) against Human Malignant Glioblastoma” J. Med. Chem. 202063, 12707-12724. DOI: 10.1021/acs.jmedchem.0c01059
  2. M. Bosco, S.-J. Paik, P. Busca, S. E. H. Moore, C. Gravier-Pelletier “Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation” Molecules 2020, 25, 4969. DOI: 10.3390/molecules25214969
  3. C. Fleurisson, E. Benedetti, L. Micouin Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications Synlett 2021, 31, 858-874. DOI: 10.1055/s-0040-1707324
  4. X. Chen, P. Coric, V. Larue, S. Turcaud, X. Wang, S. Nonin-Lecomte, S. Bouaziz “The HIV-1 maturation inhibitor, EP39, interferes with the dynamic helix-coil equilibrium of the CA-SP1 junction of Gag” Eur. J. Med. Chem.2020204, 112634 DOI: https://doi.org/10.1016/j.ejmech.2020.112634
October 2020
  1. C. Kitoun, M. Fonvielle, N. Sakkas, M. Lefresne, F. Djago, Q. Blancart Remaury, P. Poinot, M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo. “Phosphine-Mediated Bioconjugation of the 3′-end of RNA” Org. Lett., 2020, Just Acccepted.   https://doi.org/10.1021/acs.orglett.0c02982
  2. C. Aubry, P. Clerici, C. Gerbaud, L. Micouin, J.-L. Pernodet, S. Lautru, Revised structure of Anthelvencine A and characterization of the Anthelvencin Biosynthetic gene cluster.  ACS Chem Biol. 2020, 15, 945-951. https://doi.org/10.1021/acschembio.9b00960
  3. T. Zhang, L. Le Corre, O. Reinaud, B. Colasson “A Promising Approach for Controlling the 2nd Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen-Bonded Capsule” Chem. Eur. J. 2020 in press. https://doi.org/10.1002/chem.202004370.
  4. J. K. Aw, K. C. Boellaard, T. K. Tan, J. Yap, Y.P. Loh, B. Colasson, È. Blanc, Y. Lam, F. M. Fung “Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App” J. Chem. Ed. 2020, 97, 3877-3881. https://doi.org/10.1021/acs.jchemed.0c00387
July 2020
1) Dubois L, Pietrancosta N, Cabaye A, Fanget I, Debacker C, Gilormini PA, Dansette PM, Dairou J, Biot C, Froissart R, Goupil-Lamy A, Bertrand HO, Acher FC, McCort-Tranchepain I, Gasnier B, Anne C. “Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin.” J. Med. Chem. 2020  Online ahead of print.  https://doi.org/10.1021/acs.jmedchem.9b02119.  PMID: 32608236

2) H.Liu, Ping Yi, W. Zhao, Y. Wu, F. Acher, J.-P. Pin, J. Liu and P. Rondard “Illuminating the allosteric modulation of the calcium-sensing receptor” Proc Natl Acad Sci U S A 2020, 117, 21711-21722. https://doi.org/10.1073/pnas.1922231117

3) C. Atdjian, D. Coelho, L. Iannazzo , M. Ethève-Quelquejeu, E. Braud “Synthesis of Triazole-Linked SAM-Adenosine Conjugates: Functionalization of Adenosine at N-1 or N-6 Position without Protecting Groups” Molecules 2020, 25, 3241; https://doi.org/10.3390/molecules25143241

June 2020
  1. N. Babić, M. Orio, F. Peyrot. “Unexpected rapid aerobic transformation of 2,2,6,6-tetraethyl-4-oxo(piperidin-1-yloxyl) radical by cytochrome P450 in the presence of NADPH: Evidence against a simple reduction of the nitroxide moiety to the hydroxylamine”. Free Radic. Biol. Med. 2020, 156, 144-156. DOI: https://doi.org/10.1016/j.freeradbiomed.2020.05.021
  2. Kherbouche, Y. Luo, N. Félidj, C. Mangeney “Plasmon-Mediated Surface Functionalization: New Horizons for the Control of Surface Chemistry on the Nanoscale” Chem. Mater. 2020, 32, 5442. DOI: https://doi.org/10.1021/acs.chemmater.0c00921

 

Mai 2020
  1. Y. LuoY. XiaoD. OnidasL. IannazzoM. Ethève-QuelquejeuA. LamouriN. FélidjS. Mahouche-CherguiT. BruléN. Gagey-EilsteinF. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles”.  Chem. Commun., 2020, Advance Article https://doi.org/10.1039/D0CC02842H
  2. Decorbie, I. Tijunelyte, S. Gam-Derouich, J. Solard, A. Lamouri, P. Decorse, N. Felidj, C. Gauchotte-Lindsay, E. Rinnert, C. Mangeney, N. Lidgi-Guigui “Sensing Polymer/Paracetamol Interaction with an Independent Component Analysis-Based SERS-MIP Nanosensor” Plasmonics 2020, 15, 1533. DOI: https://doi.org/10.1007/s11468-020-01177-9
  3. Luo, Y. Xiao, D. Onidas, L. Iannazzo, M. Ethève-Quelquejeu, A. Lamouri, N. Félidj, S. Mahouche-Chergui, T. Brulé, N. Gagey-Eilstein, F. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles” Chem. Commun. 2020, 56, 6822. DOI: https://doi.org/10.1039/D0CC02842H
April 2020
(1) Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Diazabicyclooctane functionalization for inhibition of β-lactamases from enterobacteria”. Journal of Medicinal Chemistry, Just Accepted, https://doi.org/10.1021/acs.jmedchem.9b02125
March 2020
(1) A. Mikou, A. Cabayé, A. Goupil, H.-O. Bertrand, J.-P. Mothet, F. Acher “Asc-1 Transporter (SLC7A10): Homology models and molecular dynamics insights into the first steps of the transport mechanism.” Sci.Rep. DOI: doi.org/10.1038/s41598-020-60617-y

(2) Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, Giros B, Epelbaum J, Rosenmund C, Dutar P, Daumas S, El Mestikawy S, Pietrancosta N. “LSP5-2157 a new inhibitor of vesicular glutamate transporters.” Neuropharmacology. 2020 164 107902. doi: 10.1016/j.neuropharm.2019.107902.

January 2020
  1. Médard, P. Decorse, C. Mangeney, J. Pinson, M. Fagnoni, S. Protti “Simultaneous Photografting of Two Organic Groups on a Gold Surface by using Arylazo Sulfones as Single Precursors” Langmuir 2020, 36, 11, 2786. DOI: https://doi.org/10.1021/acs.langmuir.9b03878

 

January 2020
B. Colasson, A. Credi, B. Ventura “Photoinduced electron transfer involving a naphthalimide chromophore in switchable and flexible [2]rotaxanes“ Chem. Eur. J.202026, 534-542. doi: 10.1002/chem.201904155.
December 2019
  1. H. Habrian, J. Levitz, V. Vyklicky, Z. Fu, A.Hoagland, I. McCort-Tranchepain, F. Acher, E. Y. Isacoff “Conformational pathway provides unique sensitivity to a synaptic mGluR” Nature Commun. 2019, 10, 5572 doi:10.1038/s41467-019-13407-8
  2. Abi Fayssal, A. Giungi, F. Berhal, G. Prestat “Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes” Org. Process Res. Dev., 10.1021/acs.oprd.9b00400
November 2019
Hayek, N. Pietrancosta, A. A. Hovhannisyan, R. Alves de Sousa N. Bekaddour, L. Ermellino, E. Tramontano, S. Arnould, C. Sardet, J. Dairou, O. Diaz, V. Lotteau, S. Nisole, G. Melikyan, J.-H. Herbeuval, P.- O. Vidalain. “Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition” Eur. J. Med. Chem. DOI: 10.1016/j.ejmech.2019.111855
October 2019
Zahim, D. Ajami, P. Laurent, H. Valkenier, O. Reinaud, M. Luhmer, I. Jabin ” Synthesis and Binding Properties of a Tren-Capped Hexahomotrioxacalix[3]arene” ChemPhysChem 10.1002/cphc.201900951
September 2019

N. Babić, F. Peyrot. “New synthetic route to 2,2,6,6-tetraethylpiperidin-4-one: A key-intermediate towards tetraethyl nitroxides”. Tet. Lett. 2019, 60(44), 151207. DOI: https://doi.org/10.1016/j.tetlet.2019.151207

February 2019

N. Babić, F. Peyrot. “Molecular Probes for Evaluation of Oxidative Stress by In Vivo EPR Spectroscopy and Imaging: State-of-the-Art and Limitations”. Magnetochemistry 2019, I(1), 13. DOI: https://doi.org/10.3390/magnetochemistry5010013

june 2023

 

  1. Moreau TRJ., Bondet V., Rodero MP., Duffy D. “Heterogeneity and functions of the 13 IFN-α subtypes – lucky for some?” Eur J Immunol. 2023 Jun 27:e2250307. doi: 10.1002/eji.202250307.
  2. Fayand A., Hentgen V., Posseme C., Lacout C., Picard C., Moguelet P., Cescato M., Sbeih N., Moreau TRJ., Zhu YY., Charuel JL., Corneau A., Deibener-Kaminsky J., Dupuy S., Fusaro M., Hoareau B., Hovnanian A., Langlois V., Le Corre L., Maciel TT., Miskinyte S., Miyara M., Moulinet T., Perret M., Schuhmacher MH., Rignault-Bricard R., Viel S., Vinit A., Soria A., Duffy D., Launay JM., Callebert J., Herbeuval JP., Rodero MP., Georgin-Lavialle S. “Successful treatment of JAK1 associated inflammatory disease.” J Allergy Clin Immunol. 2023 Jun 19:S0091-6749(23)00799-6. doi: 10.1016/j.jaci.2023.06.004
  3. Bader-Meunier B., Breton S., Duffy D., Gitiaux C., Quartier P., Lemelle I., Meyer A., Welfringer-Morin A., Frémond ML., Charuel JL., Rodero MP., Melki I. “Osteonecrosis in patients with juvenile dermatomyositis: is it associated with anti-MDA5 autoantibody?” Rheumatology (Oxford). 2023 Jan 2:keac696. doi: 10.1093/rheumatology/keac696.
Mai 2023

 

  1. Le Corre L., Padovani D. “Mechanism-based and computational modeling of hydrogen sulfide biogenesis inhibition: interfacial inhibition” Scientific reports, 2023, 13, 7287. Doi: https://www.nature.com/articles/s41598-023-34405-3
  2. Coelho, D.; Le Corre, L.; Bartosik, K.; Iannazzo, L.; Braud, E.; Etheve-Quelquejeu, M. “Synthesis of Bisubstrate Analogues for RNA Methylation Studies using two Transition Metal-Catalyzed Reactions” Chem. Eur. J. 2023, e202301134.
April 2023
  1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
  2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
February 2023
  1. Flavie Bouchet, Jean-Philippe Barnier, Ines Sayah, Youcef Bagdad, Maria A. Miteva, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Ruthenium-Catalyzed Cycloaddition for Introducing Chemical Di-versity in Second generation b-Lactamase inhibitors”. ChemMedChem 2023, e202300077.
  2. Rančić A., Babić N., Orio M., Peyrot F. “Structural Features Governing the Metabolic Stability of Tetraethyl-Substituted Nitroxides in Rat Liver Microsomes”  Antioxidants, 2023, 12(2), 402. DOI:  https://doi.org/10.3390/antiox12020402
January 2023
  1. Felder, S.; Delcourt, M.-L.; Rodríguez, R.; Favereau, L.; Jeanne Crassous, J.; Micouin, L.; Benedetti, E. “Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives”, J. Mater. Chem. C 202311, 2053 DOI: https://doi.org/10.1039/D2TC04885J
  2. Galardon, E.; Mathas, N.; Padovani, D.; Le Corre, L.; Poncet, G.; Dairou, J. Persulfidation of DJ-1: Mechanism and Consequences.” Biomolecules 2023, 13, 27. DOI: https://doi.org/10.3390/biom13010027
December 2022
  1. Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein “Enzymatic synthesis of vancomycin-modified DNA”, Molecule, 2022, doi.org/10.3390/molecules27248927
October 2022
  1. C. Kitoun, S. Saidjalolov, D. Bouquet, F. Djago, Q. Blancart Remaury, B. Sargueil, P. Poinot, Pauline; M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger Ligation to Access to Stable Aminoacyl- or Peptidyl-dinucleotides” ACS Omega., 2022, just accepted.
  2. Rietmeyer, L.; Li de la Sierra-Gallay, I.; Schepers, G.; Dorchêne, D.; Iannazzo, L.; Patin, D.; Touzé, T.; van Tilbeurgh, H.; Herdewijn, P.; Etheve-Quelquejeu, M.; Fonvielle, M. “Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis” Nucleic Acids Research, 2022, just accepted
  3. S. Felder, C. Sagné, E. Benedetti, L. Micouin “Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity
    through Scaffold Hopping” ACS Chemical Biology, 2022, 17, 3069. DOI: https://doi.org/10.1021/acschembio.2c00171
August 2022

1) J.-P. Barnier, S. Saidjalolov, F. Bouchet, L. Mayer, Z. Edoo, I. Sayah, L. Iannazzo, M.e Ethève-Quelquejeu, J.-L. Mainardi, E. Braud “Modulation of the Specificity of Carbapenems and Diazabicyclooctanes for Selective Activity against Mycobacterium tuberculosis” Antimicrob. Agents Chemother. 2022, Ahead of Print

DOI: https://doi.org/10.1128/aac.02357-21

June 2022

1) F. Peyrot, S. Lajnef, D.-L. Versace. “Electron Paramagnetic Resonance Spin Trapping (EPR–ST) Technique in Photopolymerization Processes” Catalysts, 2022, 12, (7), 772; DOI: https://doi.org/10.3390/catal12070772

Mai 2022

1) V. Meynier, L. Iannazzo, M. Catala, S. Oerum, E. Braud, C.Atdjian, P. Barraud, M. Fonvielle, C. Tisné, M.Ethève-Quelquejeu “Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase” Nucleic Acids Research, 2022, 50, (10), 5793–5806. DOI: https://doi.org/10.1093/nar/gkac354

April 2022
  1. M. F. Cunha,   I.Pranke, A. Sassi, C. Schreiweis, S.  Moriceau, D. Vidovic, A. Hatton, M. S. Carlon, G. Creste, F. Berhal, G. Prestat, R. Freund, N. Odolczyk, J. P. Jais, C. Gravier-Pelletier, P.  Zielenkiewicz, V. Jullien, A. Hinzpeter, F. Oury, A. Edelman, I. Sermet-Gaudelus “Systemic Bis-Phosphinic Acid Derivative Restores Chloride Transport in Cystic Fibrosis Mice” Sci Rep 2022, 12 (1), 6132. DOI: https://doi.org/10.1038/s41598-022-09678-9.
  2. Li, K. Aubertin, D. Onidas, P. Nizard, N. Felidj, F. Gazeau, C. Mangeney, Y. Luo “Recent advances in non-plasmonic SERS nanostructures for biomedical applications” WIREs Nanomedicine & Nanobiotechnology 2022. DOI: https://doi.org/10.1002/wnan.1795
Mars 2022

1) M. Oliver, L, Le Corre, M. Poinsot, M, Bosco, H. Wan, A. Amoroso, B. Joris, A. Bouhss, S. Calvet-Vitale, C. Gravier-Pelletier “A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling” Molecules 2022, 27(6), 1769. DOI:  https://doi.org/10.3390/molecules27061769

February 2022
  1. D. Padovani, E. Galardon, “Molecular Basis for the Interaction of Catalase with d-Penicillamine: Rationalization of Some of Its Deleterious Effects” Chem. Res. Toxicol. 2022, 35, 3, 412–421 DOI: https://doi.org/10.1021/acs.chemrestox.1c00313
Janaury 2022
  1. D. R. Boyd, N. D. Sharma, P. J. Stevenson, P. Hoering, C. C. R. Allen, P. M. Dansette “Monooxygenase- and Dioxygenase-Catalyzed Oxidative Dearomatization of Thiophenes by Sulfoxidation, cis-Dihydroxylation and Epoxidation”. Int J Mol Sci. 2022, 23(2) 909. DOI:https://doi.org/10.3390/ijms23020909 
  2. Li, P. Nizard, D. Onidas, A. Lamouri, J. Pinson, S. Mahouche-Chergui, K. Aubertin, F. Gazeau, Y. Luo, C. Mangeney “SERS Tags Derived from Silver Nanoparticles and Aryl Diazonium Salts for Cell Raman Imaging” Nanoscale 2022, 14, 1452. DOI: https://doi.org/10.1039/D1NR03148A
  3. Bicyclic 5-5 systems with one ring junction nitrogen atom: Two extra heteroatoms 2:0 Benedetti, E.; Micouin, L. Reference Collection in Chemistry, Molecular Science and Chemical Engineering Wiley, 2022. Volume 11, pp 145-173. DOI:10.1016/B978-0-12-409547-2.14935-2 
December 2021
  1. S. Felder, M.-L. Delcourt, M.H.E. Bousquet, D.  Jacquemin, R. Rodríguez, L. Favereau, J. Crassous, L. Micouin, E. Benedetti “Planar chiral analogues of PRODAN based on a [2.2]paracyclophane scaffold: Synthesis and photophysical studies”. J. Org. Chem. 2021, just accepted
  2. G. Kirby, L. Grimaud, M. R. Vitale,  G. Prestat, F. Berhal “Iron(ii)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources” Green Chem., 2021,23, 9428-9432. https://doi.org/10.1039/D1GC03495B
  3. G. De Leener, D. Over, O. Reinaud, I. Jabin Turning on anion and betaine hosting by a small structural change of a biomimetic cavity: a case study” Supramol. Chem. 2021, DOI: 10.1080/10610278.2021.2011890
  4. Bitam, S.; Elbahnsi, A.; Creste, G.; Pranke, I.; Chevalier, B.; Berhal, F.; Hoffmann, B.; Servel, N.; Tondelier, D.; Hatton, A.; Moquereau, C.; Faria Da Cunha, M.; Pastor, A.; Lepissier, A.; Hinzpeter, A.; Mornon, J.-P.; Prestat, G.; Edelman, A.; Callebaut, I.; Gravier-Pelletier, C.; Sermet-Gaudelus, I. “New Insights into Structure and Function of Bis-Phosphinic Acid Derivatives and Implications for CFTR Modulation.” Sci Rep 2021, 11, 6842.
    DOI: https://doi.org/10.1038/s41598-021-83240-x
  5. Bardin, E.; Pastor, A.; Semeraro, M.; Golec, A.; Hayes, K.; Chevalier, B.; Berhal, F.; Prestat, G.; Hinzpeter, A.; Gravier-Pelletier, C.; Pranke, I.; Sermet-Gaudelus, I. “Modulators of CFTR. Updates on Clinical Development and Future Directions.” Eur. J. Med. Chem. 2021, 113195  DOI: doi.org/10.1016/j.ejmech.2021.113195
  6. Oliver, M.; Le Corre, L.; Poinsot, M.; Corio, A.; Madegard, L.; Bosco, M.; Amoroso, A.; Joris, B.; Auger, R.; Touzé, T.; Bouhss, A.; Calvet-Vitale, S.; Gravier-Pelletier, C.“Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors.”  Org. Biomol. Chem. 2021, 19(26), 5844-5866, DOI: 10.1039/D1OB00710F.
  7. Pujol C, Legrand A, Parodi L, Boucher, J.-L.; Le Corre, L. et al. “Implication of folate deficiency in CYP2U1 loss of function.” J Exp Med. 2021; 218(11):e20210846. doi: 10.1084/jem.20210846.
October 2021
  1. S. Wu, L.A. Galan, M. Roux, F. Riobe, B. Le Guennic, Y. Guyot, T. Le Bahers, L. Micouin, O. Maury, E. Benedetti “Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation” Inorg. Chem. 2021, 60, 16194−16203. DOI: https://doi.org/10.1021/acs.inorgchem.1c01986.
  2. F. Bouchet, H. Atze,  M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger ligation to introduce chemical diversity on β-lactamase inhibitors of second generation” Org. Lett.2021, just accepted
  3. Médard, X. Sun, J. Pinson, D. Li, C. Mangeney, J.-P. Michel “Electrografting and Langmuir-Blodgett: Covalently Bound Nanometer Thick Ordered Films on Graphite” Langmuir 2021, 37, 12539. DOI: https://doi.org/10.1021/acs.langmuir.1c01723
September 2021
​A. Corio, C. Gravier-Pelletier, P. Busca “Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review.” Molecules 2021, 26(18), 5467. DOI: https://doi.org/10.3390/molecules26185467
August 2021
  1. ​J. Haubrich, J. Font, R. B. Quast, A. Goupil-Lamy, P. Scholler, D. Nevoltris, F.Acher, P. Chames, P. Rondard, L. Prezeau, J.-P. Pin “A nanobody activating metabotropic glutamate receptor 4 discriminates between homo and heterodimers.” Proc. Natl. Acad. Sci. U S A 2021,
  2. Li, Y. Luo, D. Onidas, L. He, M. Jin, F. Gazeau, J. Pinson, C. Mangeney “Surface functionalization of nanomaterials by aryl diazonium salts for biomedical sciences” Adv. Colloid & Interface Science 2021, 294, 102479. DOI: https://doi.org/10.1016/j.cis.2021.102479
July 2021
  1. Xiao, J. Gateau, A. Brun, X. Shi, F. Gazeau, C. Mangeney, Y. Luo “Hybrid nano- and microgels doped with photoacoustic contrast agents for cancer theranostics” View 2021, 2:20200176. DOI: https://doi.org/10.1002/VIW.20200176
June 2021
  1. S. Felder, S. Wu, J. Brom, L. Micouin, E. Benedetti Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis”  Chirality, 2021, 33, 506-527 DOI: https://doi.org/10.1002/chir.23335
Mai 2021
  1. Kherbouche, D. McRae, T. Geronimi, F. Lagugné-Labarthet, A. Lamouri, A. Chevillot-Biraud, C. Mangeney, N. Felidj “Extending nanoscale patterning with multipolar surface plasmon resonances” Nanoscale 2021, 13, 11051. DOI: https://doi.org/10.1039/D1NR02181H
Mars 2021
  1. S. Felder, L. Micouin, E. Benedetti “Para‐functionalization of N‐substituted 4‐amino[2.2]paracyclophanes by regioselective formylation” Eur. J. Org. Chem., 2021, 4015-4018. DOI: https://doi.org/10.1002/ejoc.202100288
  2. Barosi, A. Berisha, C. Mangeney, J. Pinson, H. Dhimane, P. I. Dalko “Efficient construction of redox responsive thin polymer layer on carbon and gold for voltage-gated delivery applications” Materials Adv. 2021, 2, 2358. DOI: https://doi.org/10.1039/D1MA00022E
February 2021
  1. D.A.B. Therien, D. M. McRae, C. Mangeney, N. Félidj, F. Lagugné-Labarthet “Three-Color Plasmon-Mediated Reduction of Diazonium Salts over Metasurfaces” Nanoscale Adv. 2021, 3, 2501. DOI: https://doi.org/10.1039/D0NA00862A

January 2021
  1. Rietmeyer, N. Fix-boulier, C. Le Fournis, L. Iannazzo, C. Kitoun, D. Patin, D. Mengin-lecreulx, M. Etheve-Quelquejeu, M. Arthur, M. Fonvielle “Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus”, Nucleic Acid Res. 2021, Accepted. DOI: http://doi.org/10.1093/nar/gkaa1242
  2. S. Saidjalolov, Z. Edoo, M. Fonvielle, L. Mayer, L. Iannazzo, M. Arthur, M. Etheve-Quelquejeu, E. Braud “Synthesis of carbapenems containing peptidoglycan-mimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity” Chem. Eur. J., 2021, Accepted. DOI: http://doi.org/10.1002/chem.202004831
  3. de Sa Nogueira D, Bourdy R, Filliol D, Quessada C, McCort-Tranchepain I, Acher F, Zwiller J, Romieu P, Befort K. “LSP2-9166, an orthosteric mGlu4 and mGlu7 receptor agonist, reduces cocaine self-administration under a progressive ratio schedule in rats” Neurosci Lett. 2020, 135603 https://doi.org/10.1016/j.neulet.2020.135603
  4. K. Abbas, N. Babić, F. Peyrot. “Detection of superoxide radical in adherent living cells by electron paramagnetic resonance (EPR) spectroscopy using cyclic nitrones”. Methods Mol. Biol. 2021, 2202, 149-163. DOI: https://doi.org/10.1007/978-1-0716-0896-8_13
November 2020
  1. B. Li, Y. Li, C. Tomkiewicz-Raulet, P. Dao, D. Lietha, E. Yen-Pon, Z. Du, X. Coumoul, C. Garbay, M. Etheve-Quelquejeu, H. Chen “Design, Synthesis, and Biological Evaluation of Covalent Inhibitors of Focal Adhesion Kinase (FAK) against Human Malignant Glioblastoma” J. Med. Chem. 202063, 12707-12724. DOI: 10.1021/acs.jmedchem.0c01059
  2. M. Bosco, S.-J. Paik, P. Busca, S. E. H. Moore, C. Gravier-Pelletier “Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation” Molecules 2020, 25, 4969. DOI: 10.3390/molecules25214969
  3. C. Fleurisson, E. Benedetti, L. Micouin Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications Synlett 2021, 31, 858-874. DOI: 10.1055/s-0040-1707324
  4. X. Chen, P. Coric, V. Larue, S. Turcaud, X. Wang, S. Nonin-Lecomte, S. Bouaziz “The HIV-1 maturation inhibitor, EP39, interferes with the dynamic helix-coil equilibrium of the CA-SP1 junction of Gag” Eur. J. Med. Chem.2020204, 112634 DOI: https://doi.org/10.1016/j.ejmech.2020.112634
October 2020
  1. C. Kitoun, M. Fonvielle, N. Sakkas, M. Lefresne, F. Djago, Q. Blancart Remaury, P. Poinot, M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo. “Phosphine-Mediated Bioconjugation of the 3′-end of RNA” Org. Lett., 2020, Just Acccepted.   https://doi.org/10.1021/acs.orglett.0c02982
  2. C. Aubry, P. Clerici, C. Gerbaud, L. Micouin, J.-L. Pernodet, S. Lautru, Revised structure of Anthelvencine A and characterization of the Anthelvencin Biosynthetic gene cluster.  ACS Chem Biol. 2020, 15, 945-951. https://doi.org/10.1021/acschembio.9b00960
  3. T. Zhang, L. Le Corre, O. Reinaud, B. Colasson “A Promising Approach for Controlling the 2nd Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen-Bonded Capsule” Chem. Eur. J. 2020 in press. https://doi.org/10.1002/chem.202004370.
  4. J. K. Aw, K. C. Boellaard, T. K. Tan, J. Yap, Y.P. Loh, B. Colasson, È. Blanc, Y. Lam, F. M. Fung “Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App” J. Chem. Ed. 2020, 97, 3877-3881. https://doi.org/10.1021/acs.jchemed.0c00387
July 2020
1) Dubois L, Pietrancosta N, Cabaye A, Fanget I, Debacker C, Gilormini PA, Dansette PM, Dairou J, Biot C, Froissart R, Goupil-Lamy A, Bertrand HO, Acher FC, McCort-Tranchepain I, Gasnier B, Anne C. “Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin.” J. Med. Chem. 2020  Online ahead of print.  https://doi.org/10.1021/acs.jmedchem.9b02119.  PMID: 32608236

2) H.Liu, Ping Yi, W. Zhao, Y. Wu, F. Acher, J.-P. Pin, J. Liu and P. Rondard “Illuminating the allosteric modulation of the calcium-sensing receptor” Proc Natl Acad Sci U S A 2020, 117, 21711-21722. https://doi.org/10.1073/pnas.1922231117

3) C. Atdjian, D. Coelho, L. Iannazzo , M. Ethève-Quelquejeu, E. Braud “Synthesis of Triazole-Linked SAM-Adenosine Conjugates: Functionalization of Adenosine at N-1 or N-6 Position without Protecting Groups” Molecules 2020, 25, 3241; https://doi.org/10.3390/molecules25143241

June 2020
  1. N. Babić, M. Orio, F. Peyrot. “Unexpected rapid aerobic transformation of 2,2,6,6-tetraethyl-4-oxo(piperidin-1-yloxyl) radical by cytochrome P450 in the presence of NADPH: Evidence against a simple reduction of the nitroxide moiety to the hydroxylamine”. Free Radic. Biol. Med. 2020, 156, 144-156. DOI: https://doi.org/10.1016/j.freeradbiomed.2020.05.021
  2. Kherbouche, Y. Luo, N. Félidj, C. Mangeney “Plasmon-Mediated Surface Functionalization: New Horizons for the Control of Surface Chemistry on the Nanoscale” Chem. Mater. 2020, 32, 5442. DOI: https://doi.org/10.1021/acs.chemmater.0c00921

 

Mai 2020
  1. Y. LuoY. XiaoD. OnidasL. IannazzoM. Ethève-QuelquejeuA. LamouriN. FélidjS. Mahouche-CherguiT. BruléN. Gagey-EilsteinF. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles”.  Chem. Commun., 2020, Advance Article https://doi.org/10.1039/D0CC02842H
  2. Decorbie, I. Tijunelyte, S. Gam-Derouich, J. Solard, A. Lamouri, P. Decorse, N. Felidj, C. Gauchotte-Lindsay, E. Rinnert, C. Mangeney, N. Lidgi-Guigui “Sensing Polymer/Paracetamol Interaction with an Independent Component Analysis-Based SERS-MIP Nanosensor” Plasmonics 2020, 15, 1533. DOI: https://doi.org/10.1007/s11468-020-01177-9
  3. Luo, Y. Xiao, D. Onidas, L. Iannazzo, M. Ethève-Quelquejeu, A. Lamouri, N. Félidj, S. Mahouche-Chergui, T. Brulé, N. Gagey-Eilstein, F. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles” Chem. Commun. 2020, 56, 6822. DOI: https://doi.org/10.1039/D0CC02842H
April 2020
(1) Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Diazabicyclooctane functionalization for inhibition of β-lactamases from enterobacteria”. Journal of Medicinal Chemistry, Just Accepted, https://doi.org/10.1021/acs.jmedchem.9b02125
March 2020
(1) A. Mikou, A. Cabayé, A. Goupil, H.-O. Bertrand, J.-P. Mothet, F. Acher “Asc-1 Transporter (SLC7A10): Homology models and molecular dynamics insights into the first steps of the transport mechanism.” Sci.Rep. DOI: doi.org/10.1038/s41598-020-60617-y

(2) Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, Giros B, Epelbaum J, Rosenmund C, Dutar P, Daumas S, El Mestikawy S, Pietrancosta N. “LSP5-2157 a new inhibitor of vesicular glutamate transporters.” Neuropharmacology. 2020 164 107902. doi: 10.1016/j.neuropharm.2019.107902.

January 2020
  1. Médard, P. Decorse, C. Mangeney, J. Pinson, M. Fagnoni, S. Protti “Simultaneous Photografting of Two Organic Groups on a Gold Surface by using Arylazo Sulfones as Single Precursors” Langmuir 2020, 36, 11, 2786. DOI: https://doi.org/10.1021/acs.langmuir.9b03878

 

January 2020
B. Colasson, A. Credi, B. Ventura “Photoinduced electron transfer involving a naphthalimide chromophore in switchable and flexible [2]rotaxanes“ Chem. Eur. J.202026, 534-542. doi: 10.1002/chem.201904155.
December 2019
  1. H. Habrian, J. Levitz, V. Vyklicky, Z. Fu, A.Hoagland, I. McCort-Tranchepain, F. Acher, E. Y. Isacoff “Conformational pathway provides unique sensitivity to a synaptic mGluR” Nature Commun. 2019, 10, 5572 doi:10.1038/s41467-019-13407-8
  2. Abi Fayssal, A. Giungi, F. Berhal, G. Prestat “Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes” Org. Process Res. Dev., 10.1021/acs.oprd.9b00400
November 2019
Hayek, N. Pietrancosta, A. A. Hovhannisyan, R. Alves de Sousa N. Bekaddour, L. Ermellino, E. Tramontano, S. Arnould, C. Sardet, J. Dairou, O. Diaz, V. Lotteau, S. Nisole, G. Melikyan, J.-H. Herbeuval, P.- O. Vidalain. “Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition” Eur. J. Med. Chem. DOI: 10.1016/j.ejmech.2019.111855
October 2019
Zahim, D. Ajami, P. Laurent, H. Valkenier, O. Reinaud, M. Luhmer, I. Jabin ” Synthesis and Binding Properties of a Tren-Capped Hexahomotrioxacalix[3]arene” ChemPhysChem 10.1002/cphc.201900951
September 2019

N. Babić, F. Peyrot. “New synthetic route to 2,2,6,6-tetraethylpiperidin-4-one: A key-intermediate towards tetraethyl nitroxides”. Tet. Lett. 2019, 60(44), 151207. DOI: https://doi.org/10.1016/j.tetlet.2019.151207

February 2019

N. Babić, F. Peyrot. “Molecular Probes for Evaluation of Oxidative Stress by In Vivo EPR Spectroscopy and Imaging: State-of-the-Art and Limitations”. Magnetochemistry 2019, I(1), 13. DOI: https://doi.org/10.3390/magnetochemistry5010013

Mai 2023

 

    1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
    2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
    3. Le Corre L., Padovani D. “Mechanism-based and computational modeling of hydrogen sulfide biogenesis inhibition: interfacial inhibition” Scientific reports, 2023, 13, 7287. Doi: https://www.nature.com/articles/s41598-023-34405-3
    4. Coelho, D.; Le Corre, L.t; Bartosik, K.; Iannazzo, L.; Braud, E.; Etheve-Quelquejeu, M. “Synthesis of Bisubstrate Analogues for RNA Methylation Studies using two Transition Metal-Catalyzed Reactions” Chem. Eur. J. 2023, e202301134.
    April 2023
    1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
    2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
    February 2023
    1. Flavie Bouchet, Jean-Philippe Barnier, Ines Sayah, Youcef Bagdad, Maria A. Miteva, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Ruthenium-Catalyzed Cycloaddition for Introducing Chemical Di-versity in Second generation b-Lactamase inhibitors”. ChemMedChem 2023, e202300077.
    2. Rančić A., Babić N., Orio M., Peyrot F. “Structural Features Governing the Metabolic Stability of Tetraethyl-Substituted Nitroxides in Rat Liver Microsomes”  Antioxidants, 2023, 12(2), 402. DOI:  https://doi.org/10.3390/antiox12020402
    January 2023
    1. Felder, S.; Delcourt, M.-L.; Rodríguez, R.; Favereau, L.; Jeanne Crassous, J.; Micouin, L.; Benedetti, E. “Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives”, J. Mater. Chem. C 202311, 2053 DOI: https://doi.org/10.1039/D2TC04885J
    2. Galardon, E.; Mathas, N.; Padovani, D.; Le Corre, L.; Poncet, G.; Dairou, J. Persulfidation of DJ-1: Mechanism and Consequences.” Biomolecules 2023, 13, 27. DOI: https://doi.org/10.3390/biom13010027
    December 2022
    1. Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein “Enzymatic synthesis of vancomycin-modified DNA”, Molecule, 2022, doi.org/10.3390/molecules27248927
    October 2022
    1. C. Kitoun, S. Saidjalolov, D. Bouquet, F. Djago, Q. Blancart Remaury, B. Sargueil, P. Poinot, Pauline; M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger Ligation to Access to Stable Aminoacyl- or Peptidyl-dinucleotides” ACS Omega., 2022, just accepted.
    2. Rietmeyer, L.; Li de la Sierra-Gallay, I.; Schepers, G.; Dorchêne, D.; Iannazzo, L.; Patin, D.; Touzé, T.; van Tilbeurgh, H.; Herdewijn, P.; Etheve-Quelquejeu, M.; Fonvielle, M. “Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis” Nucleic Acids Research, 2022, just accepted
    3. S. Felder, C. Sagné, E. Benedetti, L. Micouin “Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity
      through Scaffold Hopping” ACS Chemical Biology, 2022, 17, 3069. DOI: https://doi.org/10.1021/acschembio.2c00171
    August 2022

    1) J.-P. Barnier, S. Saidjalolov, F. Bouchet, L. Mayer, Z. Edoo, I. Sayah, L. Iannazzo, M.e Ethève-Quelquejeu, J.-L. Mainardi, E. Braud “Modulation of the Specificity of Carbapenems and Diazabicyclooctanes for Selective Activity against Mycobacterium tuberculosis” Antimicrob. Agents Chemother. 2022, Ahead of Print

    DOI: https://doi.org/10.1128/aac.02357-21

    June 2022

    1) F. Peyrot, S. Lajnef, D.-L. Versace. “Electron Paramagnetic Resonance Spin Trapping (EPR–ST) Technique in Photopolymerization Processes” Catalysts, 2022, 12, (7), 772; DOI: https://doi.org/10.3390/catal12070772

    Mai 2022

    1) V. Meynier, L. Iannazzo, M. Catala, S. Oerum, E. Braud, C.Atdjian, P. Barraud, M. Fonvielle, C. Tisné, M.Ethève-Quelquejeu “Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase” Nucleic Acids Research, 2022, 50, (10), 5793–5806. DOI: https://doi.org/10.1093/nar/gkac354

    April 2022
    1. M. F. Cunha,   I.Pranke, A. Sassi, C. Schreiweis, S.  Moriceau, D. Vidovic, A. Hatton, M. S. Carlon, G. Creste, F. Berhal, G. Prestat, R. Freund, N. Odolczyk, J. P. Jais, C. Gravier-Pelletier, P.  Zielenkiewicz, V. Jullien, A. Hinzpeter, F. Oury, A. Edelman, I. Sermet-Gaudelus “Systemic Bis-Phosphinic Acid Derivative Restores Chloride Transport in Cystic Fibrosis Mice” Sci Rep 2022, 12 (1), 6132. DOI: https://doi.org/10.1038/s41598-022-09678-9.
    2. Li, K. Aubertin, D. Onidas, P. Nizard, N. Felidj, F. Gazeau, C. Mangeney, Y. Luo “Recent advances in non-plasmonic SERS nanostructures for biomedical applications” WIREs Nanomedicine & Nanobiotechnology 2022. DOI: https://doi.org/10.1002/wnan.1795
    Mars 2022

    1) M. Oliver, L, Le Corre, M. Poinsot, M, Bosco, H. Wan, A. Amoroso, B. Joris, A. Bouhss, S. Calvet-Vitale, C. Gravier-Pelletier “A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling” Molecules 2022, 27(6), 1769. DOI:  https://doi.org/10.3390/molecules27061769

    February 2022
    1. D. Padovani, E. Galardon, “Molecular Basis for the Interaction of Catalase with d-Penicillamine: Rationalization of Some of Its Deleterious Effects” Chem. Res. Toxicol. 2022, 35, 3, 412–421 DOI: https://doi.org/10.1021/acs.chemrestox.1c00313
    Janaury 2022
    1. D. R. Boyd, N. D. Sharma, P. J. Stevenson, P. Hoering, C. C. R. Allen, P. M. Dansette “Monooxygenase- and Dioxygenase-Catalyzed Oxidative Dearomatization of Thiophenes by Sulfoxidation, cis-Dihydroxylation and Epoxidation”. Int J Mol Sci. 2022, 23(2) 909. DOI:https://doi.org/10.3390/ijms23020909 
    2. Li, P. Nizard, D. Onidas, A. Lamouri, J. Pinson, S. Mahouche-Chergui, K. Aubertin, F. Gazeau, Y. Luo, C. Mangeney “SERS Tags Derived from Silver Nanoparticles and Aryl Diazonium Salts for Cell Raman Imaging” Nanoscale 2022, 14, 1452. DOI: https://doi.org/10.1039/D1NR03148A
    3. Bicyclic 5-5 systems with one ring junction nitrogen atom: Two extra heteroatoms 2:0 Benedetti, E.; Micouin, L. Reference Collection in Chemistry, Molecular Science and Chemical Engineering Wiley, 2022. Volume 11, pp 145-173. DOI:10.1016/B978-0-12-409547-2.14935-2 
    December 2021
    1. S. Felder, M.-L. Delcourt, M.H.E. Bousquet, D.  Jacquemin, R. Rodríguez, L. Favereau, J. Crassous, L. Micouin, E. Benedetti “Planar chiral analogues of PRODAN based on a [2.2]paracyclophane scaffold: Synthesis and photophysical studies”. J. Org. Chem. 2021, just accepted
    2. G. Kirby, L. Grimaud, M. R. Vitale,  G. Prestat, F. Berhal “Iron(ii)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources” Green Chem., 2021,23, 9428-9432. https://doi.org/10.1039/D1GC03495B
    3. G. De Leener, D. Over, O. Reinaud, I. Jabin Turning on anion and betaine hosting by a small structural change of a biomimetic cavity: a case study” Supramol. Chem. 2021, DOI: 10.1080/10610278.2021.2011890
    4. Bitam, S.; Elbahnsi, A.; Creste, G.; Pranke, I.; Chevalier, B.; Berhal, F.; Hoffmann, B.; Servel, N.; Tondelier, D.; Hatton, A.; Moquereau, C.; Faria Da Cunha, M.; Pastor, A.; Lepissier, A.; Hinzpeter, A.; Mornon, J.-P.; Prestat, G.; Edelman, A.; Callebaut, I.; Gravier-Pelletier, C.; Sermet-Gaudelus, I. “New Insights into Structure and Function of Bis-Phosphinic Acid Derivatives and Implications for CFTR Modulation.” Sci Rep 2021, 11, 6842.
      DOI: https://doi.org/10.1038/s41598-021-83240-x
    5. Bardin, E.; Pastor, A.; Semeraro, M.; Golec, A.; Hayes, K.; Chevalier, B.; Berhal, F.; Prestat, G.; Hinzpeter, A.; Gravier-Pelletier, C.; Pranke, I.; Sermet-Gaudelus, I. “Modulators of CFTR. Updates on Clinical Development and Future Directions.” Eur. J. Med. Chem. 2021, 113195  DOI: doi.org/10.1016/j.ejmech.2021.113195
    6. Oliver, M.; Le Corre, L.; Poinsot, M.; Corio, A.; Madegard, L.; Bosco, M.; Amoroso, A.; Joris, B.; Auger, R.; Touzé, T.; Bouhss, A.; Calvet-Vitale, S.; Gravier-Pelletier, C.“Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors.”  Org. Biomol. Chem. 2021, 19(26), 5844-5866, DOI: 10.1039/D1OB00710F.
    7. Pujol C, Legrand A, Parodi L, Boucher, J.-L.; Le Corre, L. et al. “Implication of folate deficiency in CYP2U1 loss of function.” J Exp Med. 2021; 218(11):e20210846. doi: 10.1084/jem.20210846.
    October 2021
    1. S. Wu, L.A. Galan, M. Roux, F. Riobe, B. Le Guennic, Y. Guyot, T. Le Bahers, L. Micouin, O. Maury, E. Benedetti “Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation” Inorg. Chem. 2021, 60, 16194−16203. DOI: https://doi.org/10.1021/acs.inorgchem.1c01986.
    2. F. Bouchet, H. Atze,  M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger ligation to introduce chemical diversity on β-lactamase inhibitors of second generation” Org. Lett.2021, just accepted
    3. Médard, X. Sun, J. Pinson, D. Li, C. Mangeney, J.-P. Michel “Electrografting and Langmuir-Blodgett: Covalently Bound Nanometer Thick Ordered Films on Graphite” Langmuir 2021, 37, 12539. DOI: https://doi.org/10.1021/acs.langmuir.1c01723
    September 2021
    ​A. Corio, C. Gravier-Pelletier, P. Busca “Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review.” Molecules 2021, 26(18), 5467. DOI: https://doi.org/10.3390/molecules26185467
    August 2021
    1. ​J. Haubrich, J. Font, R. B. Quast, A. Goupil-Lamy, P. Scholler, D. Nevoltris, F.Acher, P. Chames, P. Rondard, L. Prezeau, J.-P. Pin “A nanobody activating metabotropic glutamate receptor 4 discriminates between homo and heterodimers.” Proc. Natl. Acad. Sci. U S A 2021,
    2. Li, Y. Luo, D. Onidas, L. He, M. Jin, F. Gazeau, J. Pinson, C. Mangeney “Surface functionalization of nanomaterials by aryl diazonium salts for biomedical sciences” Adv. Colloid & Interface Science 2021, 294, 102479. DOI: https://doi.org/10.1016/j.cis.2021.102479
    July 2021
    1. Xiao, J. Gateau, A. Brun, X. Shi, F. Gazeau, C. Mangeney, Y. Luo “Hybrid nano- and microgels doped with photoacoustic contrast agents for cancer theranostics” View 2021, 2:20200176. DOI: https://doi.org/10.1002/VIW.20200176
    June 2021
    1. S. Felder, S. Wu, J. Brom, L. Micouin, E. Benedetti Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis”  Chirality, 2021, 33, 506-527 DOI: https://doi.org/10.1002/chir.23335
    Mai 2021
    1. Kherbouche, D. McRae, T. Geronimi, F. Lagugné-Labarthet, A. Lamouri, A. Chevillot-Biraud, C. Mangeney, N. Felidj “Extending nanoscale patterning with multipolar surface plasmon resonances” Nanoscale 2021, 13, 11051. DOI: https://doi.org/10.1039/D1NR02181H
    Mars 2021
    1. S. Felder, L. Micouin, E. Benedetti “Para‐functionalization of N‐substituted 4‐amino[2.2]paracyclophanes by regioselective formylation” Eur. J. Org. Chem., 2021, 4015-4018. DOI: https://doi.org/10.1002/ejoc.202100288
    2. Barosi, A. Berisha, C. Mangeney, J. Pinson, H. Dhimane, P. I. Dalko “Efficient construction of redox responsive thin polymer layer on carbon and gold for voltage-gated delivery applications” Materials Adv. 2021, 2, 2358. DOI: https://doi.org/10.1039/D1MA00022E
    February 2021
    1. D.A.B. Therien, D. M. McRae, C. Mangeney, N. Félidj, F. Lagugné-Labarthet “Three-Color Plasmon-Mediated Reduction of Diazonium Salts over Metasurfaces” Nanoscale Adv. 2021, 3, 2501. DOI: https://doi.org/10.1039/D0NA00862A

    January 2021
    1. Rietmeyer, N. Fix-boulier, C. Le Fournis, L. Iannazzo, C. Kitoun, D. Patin, D. Mengin-lecreulx, M. Etheve-Quelquejeu, M. Arthur, M. Fonvielle “Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus”, Nucleic Acid Res. 2021, Accepted. DOI: http://doi.org/10.1093/nar/gkaa1242
    2. S. Saidjalolov, Z. Edoo, M. Fonvielle, L. Mayer, L. Iannazzo, M. Arthur, M. Etheve-Quelquejeu, E. Braud “Synthesis of carbapenems containing peptidoglycan-mimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity” Chem. Eur. J., 2021, Accepted. DOI: http://doi.org/10.1002/chem.202004831
    3. de Sa Nogueira D, Bourdy R, Filliol D, Quessada C, McCort-Tranchepain I, Acher F, Zwiller J, Romieu P, Befort K. “LSP2-9166, an orthosteric mGlu4 and mGlu7 receptor agonist, reduces cocaine self-administration under a progressive ratio schedule in rats” Neurosci Lett. 2020, 135603 https://doi.org/10.1016/j.neulet.2020.135603
    4. K. Abbas, N. Babić, F. Peyrot. “Detection of superoxide radical in adherent living cells by electron paramagnetic resonance (EPR) spectroscopy using cyclic nitrones”. Methods Mol. Biol. 2021, 2202, 149-163. DOI: https://doi.org/10.1007/978-1-0716-0896-8_13
    November 2020
    1. B. Li, Y. Li, C. Tomkiewicz-Raulet, P. Dao, D. Lietha, E. Yen-Pon, Z. Du, X. Coumoul, C. Garbay, M. Etheve-Quelquejeu, H. Chen “Design, Synthesis, and Biological Evaluation of Covalent Inhibitors of Focal Adhesion Kinase (FAK) against Human Malignant Glioblastoma” J. Med. Chem. 202063, 12707-12724. DOI: 10.1021/acs.jmedchem.0c01059
    2. M. Bosco, S.-J. Paik, P. Busca, S. E. H. Moore, C. Gravier-Pelletier “Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation” Molecules 2020, 25, 4969. DOI: 10.3390/molecules25214969
    3. C. Fleurisson, E. Benedetti, L. Micouin Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications Synlett 2021, 31, 858-874. DOI: 10.1055/s-0040-1707324
    4. X. Chen, P. Coric, V. Larue, S. Turcaud, X. Wang, S. Nonin-Lecomte, S. Bouaziz “The HIV-1 maturation inhibitor, EP39, interferes with the dynamic helix-coil equilibrium of the CA-SP1 junction of Gag” Eur. J. Med. Chem.2020204, 112634 DOI: https://doi.org/10.1016/j.ejmech.2020.112634
    October 2020
    1. C. Kitoun, M. Fonvielle, N. Sakkas, M. Lefresne, F. Djago, Q. Blancart Remaury, P. Poinot, M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo. “Phosphine-Mediated Bioconjugation of the 3′-end of RNA” Org. Lett., 2020, Just Acccepted.   https://doi.org/10.1021/acs.orglett.0c02982
    2. C. Aubry, P. Clerici, C. Gerbaud, L. Micouin, J.-L. Pernodet, S. Lautru, Revised structure of Anthelvencine A and characterization of the Anthelvencin Biosynthetic gene cluster.  ACS Chem Biol. 2020, 15, 945-951. https://doi.org/10.1021/acschembio.9b00960
    3. T. Zhang, L. Le Corre, O. Reinaud, B. Colasson “A Promising Approach for Controlling the 2nd Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen-Bonded Capsule” Chem. Eur. J. 2020 in press. https://doi.org/10.1002/chem.202004370.
    4. J. K. Aw, K. C. Boellaard, T. K. Tan, J. Yap, Y.P. Loh, B. Colasson, È. Blanc, Y. Lam, F. M. Fung “Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App” J. Chem. Ed. 2020, 97, 3877-3881. https://doi.org/10.1021/acs.jchemed.0c00387
    July 2020
    1) Dubois L, Pietrancosta N, Cabaye A, Fanget I, Debacker C, Gilormini PA, Dansette PM, Dairou J, Biot C, Froissart R, Goupil-Lamy A, Bertrand HO, Acher FC, McCort-Tranchepain I, Gasnier B, Anne C. “Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin.” J. Med. Chem. 2020  Online ahead of print.  https://doi.org/10.1021/acs.jmedchem.9b02119.  PMID: 32608236

    2) H.Liu, Ping Yi, W. Zhao, Y. Wu, F. Acher, J.-P. Pin, J. Liu and P. Rondard “Illuminating the allosteric modulation of the calcium-sensing receptor” Proc Natl Acad Sci U S A 2020, 117, 21711-21722. https://doi.org/10.1073/pnas.1922231117

    3) C. Atdjian, D. Coelho, L. Iannazzo , M. Ethève-Quelquejeu, E. Braud “Synthesis of Triazole-Linked SAM-Adenosine Conjugates: Functionalization of Adenosine at N-1 or N-6 Position without Protecting Groups” Molecules 2020, 25, 3241; https://doi.org/10.3390/molecules25143241

    June 2020
    1. N. Babić, M. Orio, F. Peyrot. “Unexpected rapid aerobic transformation of 2,2,6,6-tetraethyl-4-oxo(piperidin-1-yloxyl) radical by cytochrome P450 in the presence of NADPH: Evidence against a simple reduction of the nitroxide moiety to the hydroxylamine”. Free Radic. Biol. Med. 2020, 156, 144-156. DOI: https://doi.org/10.1016/j.freeradbiomed.2020.05.021
    2. Kherbouche, Y. Luo, N. Félidj, C. Mangeney “Plasmon-Mediated Surface Functionalization: New Horizons for the Control of Surface Chemistry on the Nanoscale” Chem. Mater. 2020, 32, 5442. DOI: https://doi.org/10.1021/acs.chemmater.0c00921

     

    Mai 2020
    1. Y. LuoY. XiaoD. OnidasL. IannazzoM. Ethève-QuelquejeuA. LamouriN. FélidjS. Mahouche-CherguiT. BruléN. Gagey-EilsteinF. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles”.  Chem. Commun., 2020, Advance Article https://doi.org/10.1039/D0CC02842H
    2. Decorbie, I. Tijunelyte, S. Gam-Derouich, J. Solard, A. Lamouri, P. Decorse, N. Felidj, C. Gauchotte-Lindsay, E. Rinnert, C. Mangeney, N. Lidgi-Guigui “Sensing Polymer/Paracetamol Interaction with an Independent Component Analysis-Based SERS-MIP Nanosensor” Plasmonics 2020, 15, 1533. DOI: https://doi.org/10.1007/s11468-020-01177-9
    3. Luo, Y. Xiao, D. Onidas, L. Iannazzo, M. Ethève-Quelquejeu, A. Lamouri, N. Félidj, S. Mahouche-Chergui, T. Brulé, N. Gagey-Eilstein, F. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles” Chem. Commun. 2020, 56, 6822. DOI: https://doi.org/10.1039/D0CC02842H
    April 2020
    (1) Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Diazabicyclooctane functionalization for inhibition of β-lactamases from enterobacteria”. Journal of Medicinal Chemistry, Just Accepted, https://doi.org/10.1021/acs.jmedchem.9b02125
    March 2020
    (1) A. Mikou, A. Cabayé, A. Goupil, H.-O. Bertrand, J.-P. Mothet, F. Acher “Asc-1 Transporter (SLC7A10): Homology models and molecular dynamics insights into the first steps of the transport mechanism.” Sci.Rep. DOI: doi.org/10.1038/s41598-020-60617-y

    (2) Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, Giros B, Epelbaum J, Rosenmund C, Dutar P, Daumas S, El Mestikawy S, Pietrancosta N. “LSP5-2157 a new inhibitor of vesicular glutamate transporters.” Neuropharmacology. 2020 164 107902. doi: 10.1016/j.neuropharm.2019.107902.

    January 2020
    1. Médard, P. Decorse, C. Mangeney, J. Pinson, M. Fagnoni, S. Protti “Simultaneous Photografting of Two Organic Groups on a Gold Surface by using Arylazo Sulfones as Single Precursors” Langmuir 2020, 36, 11, 2786. DOI: https://doi.org/10.1021/acs.langmuir.9b03878

     

    January 2020
    B. Colasson, A. Credi, B. Ventura “Photoinduced electron transfer involving a naphthalimide chromophore in switchable and flexible [2]rotaxanes“ Chem. Eur. J.202026, 534-542. doi: 10.1002/chem.201904155.
    December 2019
    1. H. Habrian, J. Levitz, V. Vyklicky, Z. Fu, A.Hoagland, I. McCort-Tranchepain, F. Acher, E. Y. Isacoff “Conformational pathway provides unique sensitivity to a synaptic mGluR” Nature Commun. 2019, 10, 5572 doi:10.1038/s41467-019-13407-8
    2. Abi Fayssal, A. Giungi, F. Berhal, G. Prestat “Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes” Org. Process Res. Dev., 10.1021/acs.oprd.9b00400
    November 2019
    Hayek, N. Pietrancosta, A. A. Hovhannisyan, R. Alves de Sousa N. Bekaddour, L. Ermellino, E. Tramontano, S. Arnould, C. Sardet, J. Dairou, O. Diaz, V. Lotteau, S. Nisole, G. Melikyan, J.-H. Herbeuval, P.- O. Vidalain. “Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition” Eur. J. Med. Chem. DOI: 10.1016/j.ejmech.2019.111855
    October 2019
    Zahim, D. Ajami, P. Laurent, H. Valkenier, O. Reinaud, M. Luhmer, I. Jabin ” Synthesis and Binding Properties of a Tren-Capped Hexahomotrioxacalix[3]arene” ChemPhysChem 10.1002/cphc.201900951
    September 2019

    N. Babić, F. Peyrot. “New synthetic route to 2,2,6,6-tetraethylpiperidin-4-one: A key-intermediate towards tetraethyl nitroxides”. Tet. Lett. 2019, 60(44), 151207. DOI: https://doi.org/10.1016/j.tetlet.2019.151207

    February 2019

    N. Babić, F. Peyrot. “Molecular Probes for Evaluation of Oxidative Stress by In Vivo EPR Spectroscopy and Imaging: State-of-the-Art and Limitations”. Magnetochemistry 2019, I(1), 13. DOI: https://doi.org/10.3390/magnetochemistry5010013

    Mai 2023
    1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
    2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
    3. Le Corre L., Padovani D. “Mechanism-based and computational modeling of hydrogen sulfide biogenesis inhibition: interfacial inhibition” Scientific reports, 2023, 13, 7287. Doi: https://www.nature.com/articles/s41598-023-34405-3
    April 2023
    1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
    2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
    February 2023
    1. Flavie Bouchet, Jean-Philippe Barnier, Ines Sayah, Youcef Bagdad, Maria A. Miteva, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Ruthenium-Catalyzed Cycloaddition for Introducing Chemical Di-versity in Second generation b-Lactamase inhibitors”. ChemMedChem 2023, e202300077.
    2. Rančić A., Babić N., Orio M., Peyrot F. “Structural Features Governing the Metabolic Stability of Tetraethyl-Substituted Nitroxides in Rat Liver Microsomes”  Antioxidants, 2023, 12(2), 402. DOI:  https://doi.org/10.3390/antiox12020402
    January 2023
    1. Felder, S.; Delcourt, M.-L.; Rodríguez, R.; Favereau, L.; Jeanne Crassous, J.; Micouin, L.; Benedetti, E. “Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives”, J. Mater. Chem. C 202311, 2053 DOI: https://doi.org/10.1039/D2TC04885J
    2. Galardon, E.; Mathas, N.; Padovani, D.; Le Corre, L.; Poncet, G.; Dairou, J. Persulfidation of DJ-1: Mechanism and Consequences.” Biomolecules 2023, 13, 27. DOI: https://doi.org/10.3390/biom13010027
    December 2022
    1. Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein “Enzymatic synthesis of vancomycin-modified DNA”, Molecule, 2022, doi.org/10.3390/molecules27248927
    October 2022
    1. C. Kitoun, S. Saidjalolov, D. Bouquet, F. Djago, Q. Blancart Remaury, B. Sargueil, P. Poinot, Pauline; M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger Ligation to Access to Stable Aminoacyl- or Peptidyl-dinucleotides” ACS Omega., 2022, just accepted.
    2. Rietmeyer, L.; Li de la Sierra-Gallay, I.; Schepers, G.; Dorchêne, D.; Iannazzo, L.; Patin, D.; Touzé, T.; van Tilbeurgh, H.; Herdewijn, P.; Etheve-Quelquejeu, M.; Fonvielle, M. “Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis” Nucleic Acids Research, 2022, just accepted
    3. S. Felder, C. Sagné, E. Benedetti, L. Micouin “Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity
      through Scaffold Hopping” ACS Chemical Biology, 2022, 17, 3069. DOI: https://doi.org/10.1021/acschembio.2c00171
    August 2022

    1) J.-P. Barnier, S. Saidjalolov, F. Bouchet, L. Mayer, Z. Edoo, I. Sayah, L. Iannazzo, M.e Ethève-Quelquejeu, J.-L. Mainardi, E. Braud “Modulation of the Specificity of Carbapenems and Diazabicyclooctanes for Selective Activity against Mycobacterium tuberculosis” Antimicrob. Agents Chemother. 2022, Ahead of Print

    DOI: https://doi.org/10.1128/aac.02357-21

    June 2022

    1) F. Peyrot, S. Lajnef, D.-L. Versace. “Electron Paramagnetic Resonance Spin Trapping (EPR–ST) Technique in Photopolymerization Processes” Catalysts, 2022, 12, (7), 772; DOI: https://doi.org/10.3390/catal12070772

    Mai 2022

    1) V. Meynier, L. Iannazzo, M. Catala, S. Oerum, E. Braud, C.Atdjian, P. Barraud, M. Fonvielle, C. Tisné, M.Ethève-Quelquejeu “Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase” Nucleic Acids Research, 2022, 50, (10), 5793–5806. DOI: https://doi.org/10.1093/nar/gkac354

    April 2022
    1. M. F. Cunha,   I.Pranke, A. Sassi, C. Schreiweis, S.  Moriceau, D. Vidovic, A. Hatton, M. S. Carlon, G. Creste, F. Berhal, G. Prestat, R. Freund, N. Odolczyk, J. P. Jais, C. Gravier-Pelletier, P.  Zielenkiewicz, V. Jullien, A. Hinzpeter, F. Oury, A. Edelman, I. Sermet-Gaudelus “Systemic Bis-Phosphinic Acid Derivative Restores Chloride Transport in Cystic Fibrosis Mice” Sci Rep 2022, 12 (1), 6132. DOI: https://doi.org/10.1038/s41598-022-09678-9.
    2. Li, K. Aubertin, D. Onidas, P. Nizard, N. Felidj, F. Gazeau, C. Mangeney, Y. Luo “Recent advances in non-plasmonic SERS nanostructures for biomedical applications” WIREs Nanomedicine & Nanobiotechnology 2022. DOI: https://doi.org/10.1002/wnan.1795
    Mars 2022

    1) M. Oliver, L, Le Corre, M. Poinsot, M, Bosco, H. Wan, A. Amoroso, B. Joris, A. Bouhss, S. Calvet-Vitale, C. Gravier-Pelletier “A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling” Molecules 2022, 27(6), 1769. DOI:  https://doi.org/10.3390/molecules27061769

    February 2022
    1. D. Padovani, E. Galardon, “Molecular Basis for the Interaction of Catalase with d-Penicillamine: Rationalization of Some of Its Deleterious Effects” Chem. Res. Toxicol. 2022, 35, 3, 412–421 DOI: https://doi.org/10.1021/acs.chemrestox.1c00313
    Janaury 2022
    1. D. R. Boyd, N. D. Sharma, P. J. Stevenson, P. Hoering, C. C. R. Allen, P. M. Dansette “Monooxygenase- and Dioxygenase-Catalyzed Oxidative Dearomatization of Thiophenes by Sulfoxidation, cis-Dihydroxylation and Epoxidation”. Int J Mol Sci. 2022, 23(2) 909. DOI:https://doi.org/10.3390/ijms23020909 
    2. Li, P. Nizard, D. Onidas, A. Lamouri, J. Pinson, S. Mahouche-Chergui, K. Aubertin, F. Gazeau, Y. Luo, C. Mangeney “SERS Tags Derived from Silver Nanoparticles and Aryl Diazonium Salts for Cell Raman Imaging” Nanoscale 2022, 14, 1452. DOI: https://doi.org/10.1039/D1NR03148A
    3. Bicyclic 5-5 systems with one ring junction nitrogen atom: Two extra heteroatoms 2:0 Benedetti, E.; Micouin, L. Reference Collection in Chemistry, Molecular Science and Chemical Engineering Wiley, 2022. Volume 11, pp 145-173. DOI:10.1016/B978-0-12-409547-2.14935-2 
    December 2021
    1. S. Felder, M.-L. Delcourt, M.H.E. Bousquet, D.  Jacquemin, R. Rodríguez, L. Favereau, J. Crassous, L. Micouin, E. Benedetti “Planar chiral analogues of PRODAN based on a [2.2]paracyclophane scaffold: Synthesis and photophysical studies”. J. Org. Chem. 2021, just accepted
    2. G. Kirby, L. Grimaud, M. R. Vitale,  G. Prestat, F. Berhal “Iron(ii)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources” Green Chem., 2021,23, 9428-9432. https://doi.org/10.1039/D1GC03495B
    3. G. De Leener, D. Over, O. Reinaud, I. Jabin Turning on anion and betaine hosting by a small structural change of a biomimetic cavity: a case study” Supramol. Chem. 2021, DOI: 10.1080/10610278.2021.2011890
    4. Bitam, S.; Elbahnsi, A.; Creste, G.; Pranke, I.; Chevalier, B.; Berhal, F.; Hoffmann, B.; Servel, N.; Tondelier, D.; Hatton, A.; Moquereau, C.; Faria Da Cunha, M.; Pastor, A.; Lepissier, A.; Hinzpeter, A.; Mornon, J.-P.; Prestat, G.; Edelman, A.; Callebaut, I.; Gravier-Pelletier, C.; Sermet-Gaudelus, I. “New Insights into Structure and Function of Bis-Phosphinic Acid Derivatives and Implications for CFTR Modulation.” Sci Rep 2021, 11, 6842.
      DOI: https://doi.org/10.1038/s41598-021-83240-x
    5. Bardin, E.; Pastor, A.; Semeraro, M.; Golec, A.; Hayes, K.; Chevalier, B.; Berhal, F.; Prestat, G.; Hinzpeter, A.; Gravier-Pelletier, C.; Pranke, I.; Sermet-Gaudelus, I. “Modulators of CFTR. Updates on Clinical Development and Future Directions.” Eur. J. Med. Chem. 2021, 113195  DOI: doi.org/10.1016/j.ejmech.2021.113195
    6. Oliver, M.; Le Corre, L.; Poinsot, M.; Corio, A.; Madegard, L.; Bosco, M.; Amoroso, A.; Joris, B.; Auger, R.; Touzé, T.; Bouhss, A.; Calvet-Vitale, S.; Gravier-Pelletier, C.“Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors.”  Org. Biomol. Chem. 2021, 19(26), 5844-5866, DOI: 10.1039/D1OB00710F.
    7. Pujol C, Legrand A, Parodi L, Boucher, J.-L.; Le Corre, L. et al. “Implication of folate deficiency in CYP2U1 loss of function.” J Exp Med. 2021; 218(11):e20210846. doi: 10.1084/jem.20210846.
    October 2021
    1. S. Wu, L.A. Galan, M. Roux, F. Riobe, B. Le Guennic, Y. Guyot, T. Le Bahers, L. Micouin, O. Maury, E. Benedetti “Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation” Inorg. Chem. 2021, 60, 16194−16203. DOI: https://doi.org/10.1021/acs.inorgchem.1c01986.
    2. F. Bouchet, H. Atze,  M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger ligation to introduce chemical diversity on β-lactamase inhibitors of second generation” Org. Lett.2021, just accepted
    3. Médard, X. Sun, J. Pinson, D. Li, C. Mangeney, J.-P. Michel “Electrografting and Langmuir-Blodgett: Covalently Bound Nanometer Thick Ordered Films on Graphite” Langmuir 2021, 37, 12539. DOI: https://doi.org/10.1021/acs.langmuir.1c01723
    September 2021
    ​A. Corio, C. Gravier-Pelletier, P. Busca “Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review.” Molecules 2021, 26(18), 5467. DOI: https://doi.org/10.3390/molecules26185467
    August 2021
    1. ​J. Haubrich, J. Font, R. B. Quast, A. Goupil-Lamy, P. Scholler, D. Nevoltris, F.Acher, P. Chames, P. Rondard, L. Prezeau, J.-P. Pin “A nanobody activating metabotropic glutamate receptor 4 discriminates between homo and heterodimers.” Proc. Natl. Acad. Sci. U S A 2021,
    2. Li, Y. Luo, D. Onidas, L. He, M. Jin, F. Gazeau, J. Pinson, C. Mangeney “Surface functionalization of nanomaterials by aryl diazonium salts for biomedical sciences” Adv. Colloid & Interface Science 2021, 294, 102479. DOI: https://doi.org/10.1016/j.cis.2021.102479
    July 2021
    1. Xiao, J. Gateau, A. Brun, X. Shi, F. Gazeau, C. Mangeney, Y. Luo “Hybrid nano- and microgels doped with photoacoustic contrast agents for cancer theranostics” View 2021, 2:20200176. DOI: https://doi.org/10.1002/VIW.20200176
    June 2021
    1. S. Felder, S. Wu, J. Brom, L. Micouin, E. Benedetti Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis”  Chirality, 2021, 33, 506-527 DOI: https://doi.org/10.1002/chir.23335
    Mai 2021
    1. Kherbouche, D. McRae, T. Geronimi, F. Lagugné-Labarthet, A. Lamouri, A. Chevillot-Biraud, C. Mangeney, N. Felidj “Extending nanoscale patterning with multipolar surface plasmon resonances” Nanoscale 2021, 13, 11051. DOI: https://doi.org/10.1039/D1NR02181H
    Mars 2021
    1. S. Felder, L. Micouin, E. Benedetti “Para‐functionalization of N‐substituted 4‐amino[2.2]paracyclophanes by regioselective formylation” Eur. J. Org. Chem., 2021, 4015-4018. DOI: https://doi.org/10.1002/ejoc.202100288
    2. Barosi, A. Berisha, C. Mangeney, J. Pinson, H. Dhimane, P. I. Dalko “Efficient construction of redox responsive thin polymer layer on carbon and gold for voltage-gated delivery applications” Materials Adv. 2021, 2, 2358. DOI: https://doi.org/10.1039/D1MA00022E
    February 2021
    1. D.A.B. Therien, D. M. McRae, C. Mangeney, N. Félidj, F. Lagugné-Labarthet “Three-Color Plasmon-Mediated Reduction of Diazonium Salts over Metasurfaces” Nanoscale Adv. 2021, 3, 2501. DOI: https://doi.org/10.1039/D0NA00862A

    January 2021
    1. Rietmeyer, N. Fix-boulier, C. Le Fournis, L. Iannazzo, C. Kitoun, D. Patin, D. Mengin-lecreulx, M. Etheve-Quelquejeu, M. Arthur, M. Fonvielle “Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus”, Nucleic Acid Res. 2021, Accepted. DOI: http://doi.org/10.1093/nar/gkaa1242
    2. S. Saidjalolov, Z. Edoo, M. Fonvielle, L. Mayer, L. Iannazzo, M. Arthur, M. Etheve-Quelquejeu, E. Braud “Synthesis of carbapenems containing peptidoglycan-mimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity” Chem. Eur. J., 2021, Accepted. DOI: http://doi.org/10.1002/chem.202004831
    3. de Sa Nogueira D, Bourdy R, Filliol D, Quessada C, McCort-Tranchepain I, Acher F, Zwiller J, Romieu P, Befort K. “LSP2-9166, an orthosteric mGlu4 and mGlu7 receptor agonist, reduces cocaine self-administration under a progressive ratio schedule in rats” Neurosci Lett. 2020, 135603 https://doi.org/10.1016/j.neulet.2020.135603
    4. K. Abbas, N. Babić, F. Peyrot. “Detection of superoxide radical in adherent living cells by electron paramagnetic resonance (EPR) spectroscopy using cyclic nitrones”. Methods Mol. Biol. 2021, 2202, 149-163. DOI: https://doi.org/10.1007/978-1-0716-0896-8_13
    November 2020
    1. B. Li, Y. Li, C. Tomkiewicz-Raulet, P. Dao, D. Lietha, E. Yen-Pon, Z. Du, X. Coumoul, C. Garbay, M. Etheve-Quelquejeu, H. Chen “Design, Synthesis, and Biological Evaluation of Covalent Inhibitors of Focal Adhesion Kinase (FAK) against Human Malignant Glioblastoma” J. Med. Chem. 202063, 12707-12724. DOI: 10.1021/acs.jmedchem.0c01059
    2. M. Bosco, S.-J. Paik, P. Busca, S. E. H. Moore, C. Gravier-Pelletier “Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation” Molecules 2020, 25, 4969. DOI: 10.3390/molecules25214969
    3. C. Fleurisson, E. Benedetti, L. Micouin Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications Synlett 2021, 31, 858-874. DOI: 10.1055/s-0040-1707324
    4. X. Chen, P. Coric, V. Larue, S. Turcaud, X. Wang, S. Nonin-Lecomte, S. Bouaziz “The HIV-1 maturation inhibitor, EP39, interferes with the dynamic helix-coil equilibrium of the CA-SP1 junction of Gag” Eur. J. Med. Chem.2020204, 112634 DOI: https://doi.org/10.1016/j.ejmech.2020.112634
    October 2020
    1. C. Kitoun, M. Fonvielle, N. Sakkas, M. Lefresne, F. Djago, Q. Blancart Remaury, P. Poinot, M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo. “Phosphine-Mediated Bioconjugation of the 3′-end of RNA” Org. Lett., 2020, Just Acccepted.   https://doi.org/10.1021/acs.orglett.0c02982
    2. C. Aubry, P. Clerici, C. Gerbaud, L. Micouin, J.-L. Pernodet, S. Lautru, Revised structure of Anthelvencine A and characterization of the Anthelvencin Biosynthetic gene cluster.  ACS Chem Biol. 2020, 15, 945-951. https://doi.org/10.1021/acschembio.9b00960
    3. T. Zhang, L. Le Corre, O. Reinaud, B. Colasson “A Promising Approach for Controlling the 2nd Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen-Bonded Capsule” Chem. Eur. J. 2020 in press. https://doi.org/10.1002/chem.202004370.
    4. J. K. Aw, K. C. Boellaard, T. K. Tan, J. Yap, Y.P. Loh, B. Colasson, È. Blanc, Y. Lam, F. M. Fung “Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App” J. Chem. Ed. 2020, 97, 3877-3881. https://doi.org/10.1021/acs.jchemed.0c00387
    July 2020
    1) Dubois L, Pietrancosta N, Cabaye A, Fanget I, Debacker C, Gilormini PA, Dansette PM, Dairou J, Biot C, Froissart R, Goupil-Lamy A, Bertrand HO, Acher FC, McCort-Tranchepain I, Gasnier B, Anne C. “Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin.” J. Med. Chem. 2020  Online ahead of print.  https://doi.org/10.1021/acs.jmedchem.9b02119.  PMID: 32608236

    2) H.Liu, Ping Yi, W. Zhao, Y. Wu, F. Acher, J.-P. Pin, J. Liu and P. Rondard “Illuminating the allosteric modulation of the calcium-sensing receptor” Proc Natl Acad Sci U S A 2020, 117, 21711-21722. https://doi.org/10.1073/pnas.1922231117

    3) C. Atdjian, D. Coelho, L. Iannazzo , M. Ethève-Quelquejeu, E. Braud “Synthesis of Triazole-Linked SAM-Adenosine Conjugates: Functionalization of Adenosine at N-1 or N-6 Position without Protecting Groups” Molecules 2020, 25, 3241; https://doi.org/10.3390/molecules25143241

    June 2020
    1. N. Babić, M. Orio, F. Peyrot. “Unexpected rapid aerobic transformation of 2,2,6,6-tetraethyl-4-oxo(piperidin-1-yloxyl) radical by cytochrome P450 in the presence of NADPH: Evidence against a simple reduction of the nitroxide moiety to the hydroxylamine”. Free Radic. Biol. Med. 2020, 156, 144-156. DOI: https://doi.org/10.1016/j.freeradbiomed.2020.05.021
    2. Kherbouche, Y. Luo, N. Félidj, C. Mangeney “Plasmon-Mediated Surface Functionalization: New Horizons for the Control of Surface Chemistry on the Nanoscale” Chem. Mater. 2020, 32, 5442. DOI: https://doi.org/10.1021/acs.chemmater.0c00921

     

    Mai 2020
    1. Y. LuoY. XiaoD. OnidasL. IannazzoM. Ethève-QuelquejeuA. LamouriN. FélidjS. Mahouche-CherguiT. BruléN. Gagey-EilsteinF. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles”.  Chem. Commun., 2020, Advance Article https://doi.org/10.1039/D0CC02842H
    2. Decorbie, I. Tijunelyte, S. Gam-Derouich, J. Solard, A. Lamouri, P. Decorse, N. Felidj, C. Gauchotte-Lindsay, E. Rinnert, C. Mangeney, N. Lidgi-Guigui “Sensing Polymer/Paracetamol Interaction with an Independent Component Analysis-Based SERS-MIP Nanosensor” Plasmonics 2020, 15, 1533. DOI: https://doi.org/10.1007/s11468-020-01177-9
    3. Luo, Y. Xiao, D. Onidas, L. Iannazzo, M. Ethève-Quelquejeu, A. Lamouri, N. Félidj, S. Mahouche-Chergui, T. Brulé, N. Gagey-Eilstein, F. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles” Chem. Commun. 2020, 56, 6822. DOI: https://doi.org/10.1039/D0CC02842H
    April 2020
    (1) Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Diazabicyclooctane functionalization for inhibition of β-lactamases from enterobacteria”. Journal of Medicinal Chemistry, Just Accepted, https://doi.org/10.1021/acs.jmedchem.9b02125
    March 2020
    (1) A. Mikou, A. Cabayé, A. Goupil, H.-O. Bertrand, J.-P. Mothet, F. Acher “Asc-1 Transporter (SLC7A10): Homology models and molecular dynamics insights into the first steps of the transport mechanism.” Sci.Rep. DOI: doi.org/10.1038/s41598-020-60617-y

    (2) Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, Giros B, Epelbaum J, Rosenmund C, Dutar P, Daumas S, El Mestikawy S, Pietrancosta N. “LSP5-2157 a new inhibitor of vesicular glutamate transporters.” Neuropharmacology. 2020 164 107902. doi: 10.1016/j.neuropharm.2019.107902.

    January 2020
    1. Médard, P. Decorse, C. Mangeney, J. Pinson, M. Fagnoni, S. Protti “Simultaneous Photografting of Two Organic Groups on a Gold Surface by using Arylazo Sulfones as Single Precursors” Langmuir 2020, 36, 11, 2786. DOI: https://doi.org/10.1021/acs.langmuir.9b03878

     

    January 2020
    B. Colasson, A. Credi, B. Ventura “Photoinduced electron transfer involving a naphthalimide chromophore in switchable and flexible [2]rotaxanes“ Chem. Eur. J.202026, 534-542. doi: 10.1002/chem.201904155.
    December 2019
    1. H. Habrian, J. Levitz, V. Vyklicky, Z. Fu, A.Hoagland, I. McCort-Tranchepain, F. Acher, E. Y. Isacoff “Conformational pathway provides unique sensitivity to a synaptic mGluR” Nature Commun. 2019, 10, 5572 doi:10.1038/s41467-019-13407-8
    2. Abi Fayssal, A. Giungi, F. Berhal, G. Prestat “Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes” Org. Process Res. Dev., 10.1021/acs.oprd.9b00400
    November 2019
    Hayek, N. Pietrancosta, A. A. Hovhannisyan, R. Alves de Sousa N. Bekaddour, L. Ermellino, E. Tramontano, S. Arnould, C. Sardet, J. Dairou, O. Diaz, V. Lotteau, S. Nisole, G. Melikyan, J.-H. Herbeuval, P.- O. Vidalain. “Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition” Eur. J. Med. Chem. DOI: 10.1016/j.ejmech.2019.111855
    October 2019
    Zahim, D. Ajami, P. Laurent, H. Valkenier, O. Reinaud, M. Luhmer, I. Jabin ” Synthesis and Binding Properties of a Tren-Capped Hexahomotrioxacalix[3]arene” ChemPhysChem 10.1002/cphc.201900951
    September 2019

    N. Babić, F. Peyrot. “New synthetic route to 2,2,6,6-tetraethylpiperidin-4-one: A key-intermediate towards tetraethyl nitroxides”. Tet. Lett. 2019, 60(44), 151207. DOI: https://doi.org/10.1016/j.tetlet.2019.151207

    February 2019

    N. Babić, F. Peyrot. “Molecular Probes for Evaluation of Oxidative Stress by In Vivo EPR Spectroscopy and Imaging: State-of-the-Art and Limitations”. Magnetochemistry 2019, I(1), 13. DOI: https://doi.org/10.3390/magnetochemistry5010013

    Mai 2023
    1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
    2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
    3. Le Corre L., Padovani D. “Mechanism-based and computational modeling of hydrogen sulfide biogenesis inhibition: interfacial inhibition” Scientific reports, 2023, 13, 7287. Doi: https://www.nature.com/articles/s41598-023-34405-3
    April 2023
    1. Brom, J.; Maruani, A.; Micouin, L.; Benedetti, E. “Light-driven reductive cleavage of sulfonamides promoted by thiourea organophotosensitizers”. J. Org. Chem. 2023, just accepted DOI: 10.1021/acs.joc.3c00296 (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-jvdqw)
    2. Fleurisson, C.; Graidia, N.; Foricher, Y.; Benedetti, E.; Micouin, L.;  “Intramolecular Buchwald-Hartwig N-Arylation of Bicyclic Hydrazines: Practical Access to Spiro[indoline-2,3′-piperidines]”  Org. Biomol. Chem. 2023, just accepted DOI: 10.1039/D3OB00406F (Preprint ChemRxiv – DOI: 10.26434/chemrxiv-2022-rqsqc)
    February 2023
    1. Flavie Bouchet, Jean-Philippe Barnier, Ines Sayah, Youcef Bagdad, Maria A. Miteva, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Ruthenium-Catalyzed Cycloaddition for Introducing Chemical Di-versity in Second generation b-Lactamase inhibitors”. ChemMedChem 2023, e202300077.
    2. Rančić A., Babić N., Orio M., Peyrot F. “Structural Features Governing the Metabolic Stability of Tetraethyl-Substituted Nitroxides in Rat Liver Microsomes”  Antioxidants, 2023, 12(2), 402. DOI:  https://doi.org/10.3390/antiox12020402
    January 2023
    1. Felder, S.; Delcourt, M.-L.; Rodríguez, R.; Favereau, L.; Jeanne Crassous, J.; Micouin, L.; Benedetti, E. “Compact CPL emitters based on a [2.2]paracyclophane scaffold: recent developments and future perspectives”, J. Mater. Chem. C 202311, 2053 DOI: https://doi.org/10.1039/D2TC04885J
    2. Galardon, E.; Mathas, N.; Padovani, D.; Le Corre, L.; Poncet, G.; Dairou, J. Persulfidation of DJ-1: Mechanism and Consequences.” Biomolecules 2023, 13, 27. DOI: https://doi.org/10.3390/biom13010027
    December 2022
    1. Chiara Figazzolo, Frédéric Bonhomme, Saidbakhrom Saidjalolov, Mélanie Ethève-Quelquejeu, Marcel Hollenstein “Enzymatic synthesis of vancomycin-modified DNA”, Molecule, 2022, doi.org/10.3390/molecules27248927
    October 2022
    1. C. Kitoun, S. Saidjalolov, D. Bouquet, F. Djago, Q. Blancart Remaury, B. Sargueil, P. Poinot, Pauline; M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger Ligation to Access to Stable Aminoacyl- or Peptidyl-dinucleotides” ACS Omega., 2022, just accepted.
    2. Rietmeyer, L.; Li de la Sierra-Gallay, I.; Schepers, G.; Dorchêne, D.; Iannazzo, L.; Patin, D.; Touzé, T.; van Tilbeurgh, H.; Herdewijn, P.; Etheve-Quelquejeu, M.; Fonvielle, M. “Amino-acyl tXNA as inhibitors or amino acid donors in peptide synthesis” Nucleic Acids Research, 2022, just accepted
    3. S. Felder, C. Sagné, E. Benedetti, L. Micouin “Small-Molecule 3D Ligand for RNA Recognition: Tuning Selectivity
      through Scaffold Hopping” ACS Chemical Biology, 2022, 17, 3069. DOI: https://doi.org/10.1021/acschembio.2c00171
    August 2022

    1) J.-P. Barnier, S. Saidjalolov, F. Bouchet, L. Mayer, Z. Edoo, I. Sayah, L. Iannazzo, M.e Ethève-Quelquejeu, J.-L. Mainardi, E. Braud “Modulation of the Specificity of Carbapenems and Diazabicyclooctanes for Selective Activity against Mycobacterium tuberculosis” Antimicrob. Agents Chemother. 2022, Ahead of Print

    DOI: https://doi.org/10.1128/aac.02357-21

    June 2022

    1) F. Peyrot, S. Lajnef, D.-L. Versace. “Electron Paramagnetic Resonance Spin Trapping (EPR–ST) Technique in Photopolymerization Processes” Catalysts, 2022, 12, (7), 772; DOI: https://doi.org/10.3390/catal12070772

    Mai 2022

    1) V. Meynier, L. Iannazzo, M. Catala, S. Oerum, E. Braud, C.Atdjian, P. Barraud, M. Fonvielle, C. Tisné, M.Ethève-Quelquejeu “Synthesis of RNA-cofactor conjugates and structural exploration of RNA recognition by an m6A RNA methyltransferase” Nucleic Acids Research, 2022, 50, (10), 5793–5806. DOI: https://doi.org/10.1093/nar/gkac354

    April 2022
    1. M. F. Cunha,   I.Pranke, A. Sassi, C. Schreiweis, S.  Moriceau, D. Vidovic, A. Hatton, M. S. Carlon, G. Creste, F. Berhal, G. Prestat, R. Freund, N. Odolczyk, J. P. Jais, C. Gravier-Pelletier, P.  Zielenkiewicz, V. Jullien, A. Hinzpeter, F. Oury, A. Edelman, I. Sermet-Gaudelus “Systemic Bis-Phosphinic Acid Derivative Restores Chloride Transport in Cystic Fibrosis Mice” Sci Rep 2022, 12 (1), 6132. DOI: https://doi.org/10.1038/s41598-022-09678-9.
    2. Li, K. Aubertin, D. Onidas, P. Nizard, N. Felidj, F. Gazeau, C. Mangeney, Y. Luo “Recent advances in non-plasmonic SERS nanostructures for biomedical applications” WIREs Nanomedicine & Nanobiotechnology 2022. DOI: https://doi.org/10.1002/wnan.1795
    Mars 2022

    1) M. Oliver, L, Le Corre, M. Poinsot, M, Bosco, H. Wan, A. Amoroso, B. Joris, A. Bouhss, S. Calvet-Vitale, C. Gravier-Pelletier “A Sub-Micromolar MraYAA Inhibitor with an Aminoribosyl Uridine Structure and a (S,S)-Tartaric Diamide: Synthesis, Biological Evaluation and Molecular Modeling” Molecules 2022, 27(6), 1769. DOI:  https://doi.org/10.3390/molecules27061769

    February 2022
    1. D. Padovani, E. Galardon, “Molecular Basis for the Interaction of Catalase with d-Penicillamine: Rationalization of Some of Its Deleterious Effects” Chem. Res. Toxicol. 2022, 35, 3, 412–421 DOI: https://doi.org/10.1021/acs.chemrestox.1c00313
    Janaury 2022
    1. D. R. Boyd, N. D. Sharma, P. J. Stevenson, P. Hoering, C. C. R. Allen, P. M. Dansette “Monooxygenase- and Dioxygenase-Catalyzed Oxidative Dearomatization of Thiophenes by Sulfoxidation, cis-Dihydroxylation and Epoxidation”. Int J Mol Sci. 2022, 23(2) 909. DOI:https://doi.org/10.3390/ijms23020909 
    2. Li, P. Nizard, D. Onidas, A. Lamouri, J. Pinson, S. Mahouche-Chergui, K. Aubertin, F. Gazeau, Y. Luo, C. Mangeney “SERS Tags Derived from Silver Nanoparticles and Aryl Diazonium Salts for Cell Raman Imaging” Nanoscale 2022, 14, 1452. DOI: https://doi.org/10.1039/D1NR03148A
    3. Bicyclic 5-5 systems with one ring junction nitrogen atom: Two extra heteroatoms 2:0 Benedetti, E.; Micouin, L. Reference Collection in Chemistry, Molecular Science and Chemical Engineering Wiley, 2022. Volume 11, pp 145-173. DOI:10.1016/B978-0-12-409547-2.14935-2 
    December 2021
    1. S. Felder, M.-L. Delcourt, M.H.E. Bousquet, D.  Jacquemin, R. Rodríguez, L. Favereau, J. Crassous, L. Micouin, E. Benedetti “Planar chiral analogues of PRODAN based on a [2.2]paracyclophane scaffold: Synthesis and photophysical studies”. J. Org. Chem. 2021, just accepted
    2. G. Kirby, L. Grimaud, M. R. Vitale,  G. Prestat, F. Berhal “Iron(ii)-catalyzed intermolecular aziridination of alkenes employing hydroxylamine derivatives as clean nitrene sources” Green Chem., 2021,23, 9428-9432. https://doi.org/10.1039/D1GC03495B
    3. G. De Leener, D. Over, O. Reinaud, I. Jabin Turning on anion and betaine hosting by a small structural change of a biomimetic cavity: a case study” Supramol. Chem. 2021, DOI: 10.1080/10610278.2021.2011890
    4. Bitam, S.; Elbahnsi, A.; Creste, G.; Pranke, I.; Chevalier, B.; Berhal, F.; Hoffmann, B.; Servel, N.; Tondelier, D.; Hatton, A.; Moquereau, C.; Faria Da Cunha, M.; Pastor, A.; Lepissier, A.; Hinzpeter, A.; Mornon, J.-P.; Prestat, G.; Edelman, A.; Callebaut, I.; Gravier-Pelletier, C.; Sermet-Gaudelus, I. “New Insights into Structure and Function of Bis-Phosphinic Acid Derivatives and Implications for CFTR Modulation.” Sci Rep 2021, 11, 6842.
      DOI: https://doi.org/10.1038/s41598-021-83240-x
    5. Bardin, E.; Pastor, A.; Semeraro, M.; Golec, A.; Hayes, K.; Chevalier, B.; Berhal, F.; Prestat, G.; Hinzpeter, A.; Gravier-Pelletier, C.; Pranke, I.; Sermet-Gaudelus, I. “Modulators of CFTR. Updates on Clinical Development and Future Directions.” Eur. J. Med. Chem. 2021, 113195  DOI: doi.org/10.1016/j.ejmech.2021.113195
    6. Oliver, M.; Le Corre, L.; Poinsot, M.; Corio, A.; Madegard, L.; Bosco, M.; Amoroso, A.; Joris, B.; Auger, R.; Touzé, T.; Bouhss, A.; Calvet-Vitale, S.; Gravier-Pelletier, C.“Synthesis, biological evaluation and molecular modeling of urea-containing MraY inhibitors.”  Org. Biomol. Chem. 2021, 19(26), 5844-5866, DOI: 10.1039/D1OB00710F.
    7. Pujol C, Legrand A, Parodi L, Boucher, J.-L.; Le Corre, L. et al. “Implication of folate deficiency in CYP2U1 loss of function.” J Exp Med. 2021; 218(11):e20210846. doi: 10.1084/jem.20210846.
    October 2021
    1. S. Wu, L.A. Galan, M. Roux, F. Riobe, B. Le Guennic, Y. Guyot, T. Le Bahers, L. Micouin, O. Maury, E. Benedetti “Tuning the excited state properties of [2.2]paracyclophane-based antennas to ensure efficient sensitization of lanthanide ions or singlet oxygen generation” Inorg. Chem. 2021, 60, 16194−16203. DOI: https://doi.org/10.1021/acs.inorgchem.1c01986.
    2. F. Bouchet, H. Atze,  M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo “Traceless Staudinger ligation to introduce chemical diversity on β-lactamase inhibitors of second generation” Org. Lett.2021, just accepted
    3. Médard, X. Sun, J. Pinson, D. Li, C. Mangeney, J.-P. Michel “Electrografting and Langmuir-Blodgett: Covalently Bound Nanometer Thick Ordered Films on Graphite” Langmuir 2021, 37, 12539. DOI: https://doi.org/10.1021/acs.langmuir.1c01723
    September 2021
    ​A. Corio, C. Gravier-Pelletier, P. Busca “Regioselective Functionalization of Quinolines through C-H Activation: A Comprehensive Review.” Molecules 2021, 26(18), 5467. DOI: https://doi.org/10.3390/molecules26185467
    August 2021
    1. ​J. Haubrich, J. Font, R. B. Quast, A. Goupil-Lamy, P. Scholler, D. Nevoltris, F.Acher, P. Chames, P. Rondard, L. Prezeau, J.-P. Pin “A nanobody activating metabotropic glutamate receptor 4 discriminates between homo and heterodimers.” Proc. Natl. Acad. Sci. U S A 2021,
    2. Li, Y. Luo, D. Onidas, L. He, M. Jin, F. Gazeau, J. Pinson, C. Mangeney “Surface functionalization of nanomaterials by aryl diazonium salts for biomedical sciences” Adv. Colloid & Interface Science 2021, 294, 102479. DOI: https://doi.org/10.1016/j.cis.2021.102479
    July 2021
    1. Xiao, J. Gateau, A. Brun, X. Shi, F. Gazeau, C. Mangeney, Y. Luo “Hybrid nano- and microgels doped with photoacoustic contrast agents for cancer theranostics” View 2021, 2:20200176. DOI: https://doi.org/10.1002/VIW.20200176
    June 2021
    1. S. Felder, S. Wu, J. Brom, L. Micouin, E. Benedetti Enantiopure planar chiral [2.2]paracyclophanes: Synthesis and applications in asymmetric organocatalysis”  Chirality, 2021, 33, 506-527 DOI: https://doi.org/10.1002/chir.23335
    Mai 2021
    1. Kherbouche, D. McRae, T. Geronimi, F. Lagugné-Labarthet, A. Lamouri, A. Chevillot-Biraud, C. Mangeney, N. Felidj “Extending nanoscale patterning with multipolar surface plasmon resonances” Nanoscale 2021, 13, 11051. DOI: https://doi.org/10.1039/D1NR02181H
    Mars 2021
    1. S. Felder, L. Micouin, E. Benedetti “Para‐functionalization of N‐substituted 4‐amino[2.2]paracyclophanes by regioselective formylation” Eur. J. Org. Chem., 2021, 4015-4018. DOI: https://doi.org/10.1002/ejoc.202100288
    2. Barosi, A. Berisha, C. Mangeney, J. Pinson, H. Dhimane, P. I. Dalko “Efficient construction of redox responsive thin polymer layer on carbon and gold for voltage-gated delivery applications” Materials Adv. 2021, 2, 2358. DOI: https://doi.org/10.1039/D1MA00022E
    February 2021
    1. D.A.B. Therien, D. M. McRae, C. Mangeney, N. Félidj, F. Lagugné-Labarthet “Three-Color Plasmon-Mediated Reduction of Diazonium Salts over Metasurfaces” Nanoscale Adv. 2021, 3, 2501. DOI: https://doi.org/10.1039/D0NA00862A

    January 2021
    1. Rietmeyer, N. Fix-boulier, C. Le Fournis, L. Iannazzo, C. Kitoun, D. Patin, D. Mengin-lecreulx, M. Etheve-Quelquejeu, M. Arthur, M. Fonvielle “Partition of tRNAGly isoacceptors between protein and cell-wall peptidoglycan synthesis in Staphylococcus aureus”, Nucleic Acid Res. 2021, Accepted. DOI: http://doi.org/10.1093/nar/gkaa1242
    2. S. Saidjalolov, Z. Edoo, M. Fonvielle, L. Mayer, L. Iannazzo, M. Arthur, M. Etheve-Quelquejeu, E. Braud “Synthesis of carbapenems containing peptidoglycan-mimetics and inhibition of the cross-linking activity of a transpeptidase of the L,D specificity” Chem. Eur. J., 2021, Accepted. DOI: http://doi.org/10.1002/chem.202004831
    3. de Sa Nogueira D, Bourdy R, Filliol D, Quessada C, McCort-Tranchepain I, Acher F, Zwiller J, Romieu P, Befort K. “LSP2-9166, an orthosteric mGlu4 and mGlu7 receptor agonist, reduces cocaine self-administration under a progressive ratio schedule in rats” Neurosci Lett. 2020, 135603 https://doi.org/10.1016/j.neulet.2020.135603
    4. K. Abbas, N. Babić, F. Peyrot. “Detection of superoxide radical in adherent living cells by electron paramagnetic resonance (EPR) spectroscopy using cyclic nitrones”. Methods Mol. Biol. 2021, 2202, 149-163. DOI: https://doi.org/10.1007/978-1-0716-0896-8_13
    November 2020
    1. B. Li, Y. Li, C. Tomkiewicz-Raulet, P. Dao, D. Lietha, E. Yen-Pon, Z. Du, X. Coumoul, C. Garbay, M. Etheve-Quelquejeu, H. Chen “Design, Synthesis, and Biological Evaluation of Covalent Inhibitors of Focal Adhesion Kinase (FAK) against Human Malignant Glioblastoma” J. Med. Chem. 202063, 12707-12724. DOI: 10.1021/acs.jmedchem.0c01059
    2. M. Bosco, S.-J. Paik, P. Busca, S. E. H. Moore, C. Gravier-Pelletier “Synthetic Route to Glycosyl β-1C-(phosphino)-phosphonates as Unprecedented Stable Glycosyl Diphosphate Analogs and Their Preliminary Biological Evaluation” Molecules 2020, 25, 4969. DOI: 10.3390/molecules25214969
    3. C. Fleurisson, E. Benedetti, L. Micouin Cyclic cis-1,3-Diamines Derived from Bicyclic Hydrazines: Synthesis and Applications Synlett 2021, 31, 858-874. DOI: 10.1055/s-0040-1707324
    4. X. Chen, P. Coric, V. Larue, S. Turcaud, X. Wang, S. Nonin-Lecomte, S. Bouaziz “The HIV-1 maturation inhibitor, EP39, interferes with the dynamic helix-coil equilibrium of the CA-SP1 junction of Gag” Eur. J. Med. Chem.2020204, 112634 DOI: https://doi.org/10.1016/j.ejmech.2020.112634
    October 2020
    1. C. Kitoun, M. Fonvielle, N. Sakkas, M. Lefresne, F. Djago, Q. Blancart Remaury, P. Poinot, M. Arthur, M. Etheve-Quelquejeu, L. Iannazzo. “Phosphine-Mediated Bioconjugation of the 3′-end of RNA” Org. Lett., 2020, Just Acccepted.   https://doi.org/10.1021/acs.orglett.0c02982
    2. C. Aubry, P. Clerici, C. Gerbaud, L. Micouin, J.-L. Pernodet, S. Lautru, Revised structure of Anthelvencine A and characterization of the Anthelvencin Biosynthetic gene cluster.  ACS Chem Biol. 2020, 15, 945-951. https://doi.org/10.1021/acschembio.9b00960
    3. T. Zhang, L. Le Corre, O. Reinaud, B. Colasson “A Promising Approach for Controlling the 2nd Coordination Sphere of Biomimetic Metal Complexes: Encapsulation in a Dynamic Hydrogen-Bonded Capsule” Chem. Eur. J. 2020 in press. https://doi.org/10.1002/chem.202004370.
    4. J. K. Aw, K. C. Boellaard, T. K. Tan, J. Yap, Y.P. Loh, B. Colasson, È. Blanc, Y. Lam, F. M. Fung “Interacting with Three-Dimensional Molecular Structures Using an Augmented Reality Mobile App” J. Chem. Ed. 2020, 97, 3877-3881. https://doi.org/10.1021/acs.jchemed.0c00387
    July 2020
    1) Dubois L, Pietrancosta N, Cabaye A, Fanget I, Debacker C, Gilormini PA, Dansette PM, Dairou J, Biot C, Froissart R, Goupil-Lamy A, Bertrand HO, Acher FC, McCort-Tranchepain I, Gasnier B, Anne C. “Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin.” J. Med. Chem. 2020  Online ahead of print.  https://doi.org/10.1021/acs.jmedchem.9b02119.  PMID: 32608236

    2) H.Liu, Ping Yi, W. Zhao, Y. Wu, F. Acher, J.-P. Pin, J. Liu and P. Rondard “Illuminating the allosteric modulation of the calcium-sensing receptor” Proc Natl Acad Sci U S A 2020, 117, 21711-21722. https://doi.org/10.1073/pnas.1922231117

    3) C. Atdjian, D. Coelho, L. Iannazzo , M. Ethève-Quelquejeu, E. Braud “Synthesis of Triazole-Linked SAM-Adenosine Conjugates: Functionalization of Adenosine at N-1 or N-6 Position without Protecting Groups” Molecules 2020, 25, 3241; https://doi.org/10.3390/molecules25143241

    June 2020
    1. N. Babić, M. Orio, F. Peyrot. “Unexpected rapid aerobic transformation of 2,2,6,6-tetraethyl-4-oxo(piperidin-1-yloxyl) radical by cytochrome P450 in the presence of NADPH: Evidence against a simple reduction of the nitroxide moiety to the hydroxylamine”. Free Radic. Biol. Med. 2020, 156, 144-156. DOI: https://doi.org/10.1016/j.freeradbiomed.2020.05.021
    2. Kherbouche, Y. Luo, N. Félidj, C. Mangeney “Plasmon-Mediated Surface Functionalization: New Horizons for the Control of Surface Chemistry on the Nanoscale” Chem. Mater. 2020, 32, 5442. DOI: https://doi.org/10.1021/acs.chemmater.0c00921

     

    Mai 2020
    1. Y. LuoY. XiaoD. OnidasL. IannazzoM. Ethève-QuelquejeuA. LamouriN. FélidjS. Mahouche-CherguiT. BruléN. Gagey-EilsteinF. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles”.  Chem. Commun., 2020, Advance Article https://doi.org/10.1039/D0CC02842H
    2. Decorbie, I. Tijunelyte, S. Gam-Derouich, J. Solard, A. Lamouri, P. Decorse, N. Felidj, C. Gauchotte-Lindsay, E. Rinnert, C. Mangeney, N. Lidgi-Guigui “Sensing Polymer/Paracetamol Interaction with an Independent Component Analysis-Based SERS-MIP Nanosensor” Plasmonics 2020, 15, 1533. DOI: https://doi.org/10.1007/s11468-020-01177-9
    3. Luo, Y. Xiao, D. Onidas, L. Iannazzo, M. Ethève-Quelquejeu, A. Lamouri, N. Félidj, S. Mahouche-Chergui, T. Brulé, N. Gagey-Eilstein, F. Gazeau, C. Mangeney “Raman reporters derived from aryl diazonium salts for SERS encoded-nanoparticles” Chem. Commun. 2020, 56, 6822. DOI: https://doi.org/10.1039/D0CC02842H
    April 2020
    (1) Flavie Bouchet, Heiner Atze, Matthieu Fonvielle, Zainab Edoo, Michel Arthur, Mélanie Ethève-Quelquejeu, Laura Iannazzo “Diazabicyclooctane functionalization for inhibition of β-lactamases from enterobacteria”. Journal of Medicinal Chemistry, Just Accepted, https://doi.org/10.1021/acs.jmedchem.9b02125
    March 2020
    (1) A. Mikou, A. Cabayé, A. Goupil, H.-O. Bertrand, J.-P. Mothet, F. Acher “Asc-1 Transporter (SLC7A10): Homology models and molecular dynamics insights into the first steps of the transport mechanism.” Sci.Rep. DOI: doi.org/10.1038/s41598-020-60617-y

    (2) Poirel O, Mamer LE, Herman MA, Arnulf-Kempcke M, Kervern M, Potier B, Miot S, Wang J, Favre-Besse FC, Brabet I, Laras Y, Bertrand HO, Acher F, Pin JP, Puel JL, Giros B, Epelbaum J, Rosenmund C, Dutar P, Daumas S, El Mestikawy S, Pietrancosta N. “LSP5-2157 a new inhibitor of vesicular glutamate transporters.” Neuropharmacology. 2020 164 107902. doi: 10.1016/j.neuropharm.2019.107902.

    January 2020
    1. Médard, P. Decorse, C. Mangeney, J. Pinson, M. Fagnoni, S. Protti “Simultaneous Photografting of Two Organic Groups on a Gold Surface by using Arylazo Sulfones as Single Precursors” Langmuir 2020, 36, 11, 2786. DOI: https://doi.org/10.1021/acs.langmuir.9b03878

     

    January 2020
    B. Colasson, A. Credi, B. Ventura “Photoinduced electron transfer involving a naphthalimide chromophore in switchable and flexible [2]rotaxanes“ Chem. Eur. J.202026, 534-542. doi: 10.1002/chem.201904155.
    December 2019
    1. H. Habrian, J. Levitz, V. Vyklicky, Z. Fu, A.Hoagland, I. McCort-Tranchepain, F. Acher, E. Y. Isacoff “Conformational pathway provides unique sensitivity to a synaptic mGluR” Nature Commun. 2019, 10, 5572 doi:10.1038/s41467-019-13407-8
    2. Abi Fayssal, A. Giungi, F. Berhal, G. Prestat “Iron-Catalyzed Intra-intermolecular Aminoazidation of Alkenes” Org. Process Res. Dev., 10.1021/acs.oprd.9b00400
    November 2019
    Hayek, N. Pietrancosta, A. A. Hovhannisyan, R. Alves de Sousa N. Bekaddour, L. Ermellino, E. Tramontano, S. Arnould, C. Sardet, J. Dairou, O. Diaz, V. Lotteau, S. Nisole, G. Melikyan, J.-H. Herbeuval, P.- O. Vidalain. “Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition” Eur. J. Med. Chem. DOI: 10.1016/j.ejmech.2019.111855
    October 2019
    Zahim, D. Ajami, P. Laurent, H. Valkenier, O. Reinaud, M. Luhmer, I. Jabin ” Synthesis and Binding Properties of a Tren-Capped Hexahomotrioxacalix[3]arene” ChemPhysChem 10.1002/cphc.201900951
    September 2019

    N. Babić, F. Peyrot. “New synthetic route to 2,2,6,6-tetraethylpiperidin-4-one: A key-intermediate towards tetraethyl nitroxides”. Tet. Lett. 2019, 60(44), 151207. DOI: https://doi.org/10.1016/j.tetlet.2019.151207

    February 2019

    N. Babić, F. Peyrot. “Molecular Probes for Evaluation of Oxidative Stress by In Vivo EPR Spectroscopy and Imaging: State-of-the-Art and Limitations”. Magnetochemistry 2019, I(1), 13. DOI: https://doi.org/10.3390/magnetochemistry5010013